SCHEMBL9111169

SCHEMBL9111169

CCOC(=O)CC1C=CN(C(=O)OC)C=C1Br

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ALDH1A1 P00352 6/20 0.33
KMT2A Q03164 4/20 0.33
MAPT P10636 2/20 0.33
HPGD P15428 1/20 0.33
MGAM O43451 1/20 0.33
GAA P10253 1/20 0.33
SI P14410 1/20 0.33
MGAM2 Q2M2H8 1/20 0.33
IDO1 P14902 1/20 0.32
GSK3A P49840 1/20 0.31
GSK3B P49841 1/20 0.31
TRPA1 O75762 1/20 0.31
CYP1A2 P05177 2/20 0.30
MEN1 O00255 2/20 0.30
CYP2C19 P33261 1/20 0.30
PKM P14618 1/20 0.30
MAPK1 P28482 1/20 0.30
BRD4 O60885 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9111764 0.83 TSHR (0.33) TSHRHSD17B10ALDH1A1KMT2AMAPT
SCHEMBL13413685 0.71 LPO (0.33) TSHRHSD17B10ALDH1A1HPGD
SCHEMBL19838577 0.69 HTT (0.38) HSD17B10ALDH1A1KMT2AMAPTHPGD
SCHEMBL9110269 0.68 ALDH1A1 (0.35) TSHRHSD17B10ALDH1A1KMT2AMAPT
SCHEMBL9112483 0.64 MGAM (0.36) TSHRHSD17B10ALDH1A1KMT2AMAPT
SCHEMBL6924804 0.62 GSK3A (0.41) TSHRHSD17B10ALDH1A1KMT2AMGAM
SCHEMBL736634 0.61 GSK3A (0.40) TSHRHSD17B10ALDH1A1KMT2AMAPT
SCHEMBL31598498 0.56 GSK3A (0.35) TSHRHSD17B10ALDH1A1KMT2AMAPT
SCHEMBL1649446 0.56 TSHR (0.33) TSHRCYP2C19
SCHEMBL6943189 0.56 ALDH1A1 (0.30) TSHRALDH1A1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995010505-A1 FUNCTIONALIZATION OF ACYL PYRIDINIUM SALTS SYNAPTIC PHARMACEUTICAL CORPORATION (US) 1995-04-20 WO disclosed