SCHEMBL9116097

SCHEMBL9116097

O=C(c1ccc(F)cc1F)C1CCN(CCCc2coc3ccc(Cl)cc3c2=O)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.51
KDM4E B2RXH2 1/20 0.51
KCNH2 Q12809 3/20 0.44
HSD17B10 Q99714 1/20 0.43
DRD2 P14416 2/20 0.40
GAA P10253 1/20 0.39
CHRM2 P08172 1/20 0.39
CHRM4 P08173 1/20 0.39
CHRM5 P08912 1/20 0.39
CHRM1 P11229 1/20 0.39
CHRM3 P20309 1/20 0.39
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
MAOB P27338 2/20 0.38
HRH3 Q9Y5N1 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9289676 0.89 KDM4E (0.53) ALDH1A1KDM4EHSD17B10HTR2AHTR2C
SCHEMBL9118514 0.86 HTR2A (0.53) ALDH1A1KDM4EHTR2AHTR2C
SCHEMBL9116840 0.85 KCNH2 (0.45) KCNH2DRD2CHRM2CHRM4CHRM5
SCHEMBL9117274 0.83 ALDH1A1 (0.54) ALDH1A1KDM4EKCNH2HSD17B10MEN1
SCHEMBL9117345 0.83 CHRM2 (0.49) ALDH1A1KDM4EKCNH2CHRM2CHRM4
SCHEMBL9115603 0.81 HTR2A (0.57) KDM4EHTR2AHTR2C
SCHEMBL9117523 0.79 HTR2A (0.50) KDM4EHTR2AHTR2C
SCHEMBL9116862 0.77 HTR2C (0.57) KDM4EDRD2MEN1KMT2AHTR2A
SCHEMBL9114665 0.76 DRD2 (0.49) ALDH1A1KDM4EDRD2HTR2AHTR2C
SCHEMBL9115113 0.76 HTR2A (0.53) ALDH1A1KDM4EKCNH2HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995025731-A1 NOVEL 3-(φ-(4-BENZOYLPIPERIDINO)ALKYL)-4H-BENZOPYRAN-4-ONES, PREPARATION AND THERAPEUTICAL USE THEREOF PIERRE FABRE MEDICAMENT (FR) 1995-09-28 WO claimed
WO-1995025731-A1 NOVEL 3-(φ-(4-BENZOYLPIPERIDINO)ALKYL)-4H-BENZOPYRAN-4-ONES, PREPARATION AND THERAPEUTICAL USE THEREOF PIERRE FABRE MEDICAMENT (FR) 1995-09-28 WO disclosed