SCHEMBL9117345

SCHEMBL9117345

COc1ccc2c(=O)c(CCCN3CCC(C(=O)c4ccc(F)cc4F)CC3)coc2c1

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.49
CHRM4 P08173 1/20 0.49
CHRM5 P08912 1/20 0.49
CHRM1 P11229 1/20 0.49
CHRM3 P20309 1/20 0.49
DRD4 P21917 1/20 0.49
DRD3 P35462 1/20 0.49
SIGMAR1 Q99720 1/20 0.49
KCNH2 Q12809 1/20 0.48
CPS1 P31327 1/20 0.46
MAOB P27338 2/20 0.44
HRH3 Q9Y5N1 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.41
HTR1A P08908 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9116840 0.89 KCNH2 (0.45) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL9116078 0.87 HTR2A (0.51) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL9117040 0.84 MAOB (0.51) KCNH2MAOBHRH3KDM4EALDH1A1
SCHEMBL9114665 0.83 DRD2 (0.49) KDM4EALDH1A1
SCHEMBL9116097 0.83 ALDH1A1 (0.51) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL9115981 0.80 HTR2A (0.50) KDM4EALDH1A1
SCHEMBL9115963 0.80 HTR2A (0.50) KDM4EALDH1A1
SCHEMBL9115835 0.80 HTR2A (0.50) KDM4EALDH1A1
SCHEMBL9115680 0.78 HTR2A (0.49) KDM4E
SCHEMBL9117585 0.77 HTR2A (0.51) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995025731-A1 NOVEL 3-(φ-(4-BENZOYLPIPERIDINO)ALKYL)-4H-BENZOPYRAN-4-ONES, PREPARATION AND THERAPEUTICAL USE THEREOF PIERRE FABRE MEDICAMENT (FR) 1995-09-28 WO claimed
WO-1995025731-A1 NOVEL 3-(φ-(4-BENZOYLPIPERIDINO)ALKYL)-4H-BENZOPYRAN-4-ONES, PREPARATION AND THERAPEUTICAL USE THEREOF PIERRE FABRE MEDICAMENT (FR) 1995-09-28 WO disclosed