SCHEMBL9124791

SCHEMBL9124791

COc1ccc(COc2cccnc2NC(N)=Nc2ccc(Cl)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
PPIA P62937 9/20 0.50
MAPT P10636 2/20 0.44
KDM4E B2RXH2 2/20 0.44
GAA P10253 2/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.44
SIGMAR1 Q99720 1/20 0.41
PPIF P30405 1/20 0.41
ALDH1A1 P00352 2/20 0.40
C5AR1 P21730 1/20 0.40
CRHBP P24387 1/20 0.40
CRHR2 Q13324 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9122341 0.91 PPIA (0.51) PPIASIGMAR1PPIFC5AR1
SCHEMBL9128504 0.90 NPC1 (0.54) NPC1RAB9APPIAC5AR1
SCHEMBL9125077 0.89 PPIA (0.62) PPIAPPIFC5AR1
SCHEMBL9125087 0.89 PPIA (0.59) NPC1RAB9APPIAMAPTKMT2A
SCHEMBL9126099 0.86 PPIF (0.41) NPC1RAB9APPIAMAPTKDM4E
SCHEMBL9127905 0.82 PPIA (0.45) PPIASIGMAR1PPIFALDH1A1
SCHEMBL9126127 0.81 PPIA (0.45) RAB9APPIAMAPTSIGMAR1PPIF
SCHEMBL2783284 0.81 PPIA (0.58) PPIAPPIF
SCHEMBL9124960 0.81 PPIA (0.47) PPIAMAPTKDM4EGAASIGMAR1
SCHEMBL9125102 0.80 PPIA (0.42) RAB9APPIAMAPTSIGMAR1PPIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5409943-A [(alkoxy)pyridinyl]amine compounds which are useful in the treatment of gastrointestinal disorders SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1995-04-25 US disclosed
EP-0625143-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1994-11-23 EP disclosed
WO-1993015055-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1993-08-05 WO disclosed