SCHEMBL9122341

SCHEMBL9122341

Cc1ccc(COc2cccnc2NC(N)=Nc2ccc(Cl)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PPIA P62937 12/20 0.51
SCN2A Q99250 1/20 0.42
SIGMAR1 Q99720 2/20 0.42
PPIF P30405 1/20 0.41
GRIN2D O15399 1/20 0.41
GRIN3B O60391 1/20 0.41
GRIN1 Q05586 1/20 0.41
GRIN2A Q12879 1/20 0.41
GRIN2B Q13224 1/20 0.41
GRIN2C Q14957 1/20 0.41
GRIN3A Q8TCU5 1/20 0.41
ACHE P22303 1/20 0.39
FURIN P09958 1/20 0.39
C5AR1 P21730 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9124791 0.91 NPC1 (0.51) PPIASIGMAR1PPIFC5AR1
SCHEMBL9125087 0.90 PPIA (0.59) PPIAPPIFFURINC5AR1
SCHEMBL9125077 0.90 PPIA (0.62) PPIAPPIFC5AR1
SCHEMBL9125102 0.85 PPIA (0.42) PPIASIGMAR1PPIFGRIN2DGRIN3B
SCHEMBL9126127 0.84 PPIA (0.45) PPIASIGMAR1PPIF
SCHEMBL9127905 0.83 PPIA (0.45) PPIASIGMAR1PPIF
SCHEMBL2783284 0.82 PPIA (0.58) PPIAPPIF
SCHEMBL9124960 0.82 PPIA (0.47) PPIASIGMAR1PPIF
SCHEMBL9123963 0.81 SGMS2 (0.44) PPIASIGMAR1PPIFGRIN2DGRIN3B
SCHEMBL9125719 0.81 PPIA (0.40) PPIASIGMAR1PPIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5409943-A [(alkoxy)pyridinyl]amine compounds which are useful in the treatment of gastrointestinal disorders SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1995-04-25 US disclosed
EP-0625143-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1994-11-23 EP disclosed
WO-1993015055-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1993-08-05 WO disclosed