SCHEMBL9125719

SCHEMBL9125719

Cc1cccc(COc2cccnc2NC(N)=Nc2ccc(Cl)cc2)c1F

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PPIA P62937 5/20 0.40
PPIF P30405 1/20 0.40
SIGMAR1 Q99720 1/20 0.39
GCK P35557 1/20 0.37
SGMS2 Q8NHU3 4/20 0.36
RAB9A P51151 1/20 0.36
L3MBTL1 Q9Y468 3/20 0.36
HTT P42858 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
MAPT P10636 1/20 0.34
MRGPRX4 Q96LA9 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
ALOX12 P18054 1/20 0.34
KMT2A Q03164 1/20 0.34
SGMS1 Q86VZ5 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9125354 0.90 SGMS2 (0.46) PPIAPPIFSIGMAR1SGMS2MRGPRX4
SCHEMBL9126127 0.90 PPIA (0.45) PPIAPPIFSIGMAR1GCKSGMS2
SCHEMBL9124960 0.84 PPIA (0.47) PPIAPPIFSIGMAR1SGMS2MAPT
SCHEMBL9124036 0.83 PPIF (0.48) PPIAPPIFSIGMAR1SGMS2TDP1
SCHEMBL9124709 0.82 PPIA (0.44) PPIAPPIFSIGMAR1
SCHEMBL9128712 0.82 PPIA (0.43) PPIAPPIFSIGMAR1SGMS2NPSR1
SCHEMBL9123653 0.81 SGMS2 (0.44) PPIASIGMAR1GCKSGMS2L3MBTL1
SCHEMBL9123692 0.81 PPIA (0.49) PPIAPPIFSGMS2RAB9AL3MBTL1
SCHEMBL9125102 0.81 PPIA (0.42) PPIAPPIFSIGMAR1SGMS2RAB9A
SCHEMBL9122341 0.81 PPIA (0.51) PPIAPPIFSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5409943-A [(alkoxy)pyridinyl]amine compounds which are useful in the treatment of gastrointestinal disorders SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1995-04-25 US disclosed
EP-0625143-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1994-11-23 EP disclosed
WO-1993015055-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1993-08-05 WO disclosed