SCHEMBL9128712

SCHEMBL9128712

NC(=Nc1ccc(Cl)cc1)Nc1ncccc1OCc1c(F)ccc(F)c1F

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PPIA P62937 10/20 0.43
PPIF P30405 1/20 0.43
SIGMAR1 Q99720 2/20 0.36
ADRA2A P08913 1/20 0.36
SGMS2 Q8NHU3 1/20 0.35
ALDH1A1 P00352 1/20 0.34
AR P10275 1/20 0.34
KCNH2 Q12809 1/20 0.34
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9124036 0.93 PPIF (0.48) PPIAPPIFSIGMAR1SGMS2ALDH1A1
SCHEMBL9127446 0.90 SGMS2 (0.46) PPIAPPIFSIGMAR1SGMS2ALDH1A1
SCHEMBL9127905 0.86 PPIA (0.45) PPIAPPIFSIGMAR1SGMS2ALDH1A1
SCHEMBL9129022 0.84 SGMS2 (0.46) PPIAPPIFSGMS2ALDH1A1
SCHEMBL9125354 0.84 SGMS2 (0.46) PPIAPPIFSIGMAR1SGMS2ALDH1A1
SCHEMBL9124709 0.84 PPIA (0.44) PPIAPPIFSIGMAR1
SCHEMBL9125077 0.83 PPIA (0.62) PPIAPPIF
SCHEMBL9126733 0.82 SGMS2 (0.48) PPIAPPIFSGMS2ALDH1A1
SCHEMBL9125102 0.82 PPIA (0.42) PPIAPPIFSIGMAR1SGMS2ALDH1A1
SCHEMBL9123963 0.82 SGMS2 (0.44) PPIAPPIFSIGMAR1SGMS2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5409943-A [(alkoxy)pyridinyl]amine compounds which are useful in the treatment of gastrointestinal disorders SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1995-04-25 US disclosed
EP-0625143-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1994-11-23 EP disclosed
WO-1993015055-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1993-08-05 WO disclosed