SCHEMBL9124709

SCHEMBL9124709

NC(=Nc1ccc(Cl)cc1)Nc1ncccc1OCc1ccc(F)cc1F

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PPIA P62937 4/20 0.44
PPIF P30405 1/20 0.43
PTGER1 P34995 5/20 0.42
CCR5 P51681 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
MAPK14 Q16539 3/20 0.37
CNR1 P21554 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9126099 0.90 PPIF (0.41) PPIAPPIFSIGMAR1
SCHEMBL9124036 0.85 PPIF (0.48) PPIAPPIFSIGMAR1
SCHEMBL9127446 0.84 SGMS2 (0.46) PPIAPPIFSIGMAR1
SCHEMBL9125354 0.84 SGMS2 (0.46) PPIAPPIFSIGMAR1
SCHEMBL9128712 0.84 PPIA (0.43) PPIAPPIFSIGMAR1
SCHEMBL9124960 0.83 PPIA (0.47) PPIAPPIFSIGMAR1
SCHEMBL9125719 0.82 PPIA (0.40) PPIAPPIFSIGMAR1
SCHEMBL9127905 0.82 PPIA (0.45) PPIAPPIFSIGMAR1
SCHEMBL9126127 0.82 PPIA (0.45) PPIAPPIFSIGMAR1
SCHEMBL9125077 0.81 PPIA (0.62) PPIAPPIFMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5409943-A [(alkoxy)pyridinyl]amine compounds which are useful in the treatment of gastrointestinal disorders SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1995-04-25 US disclosed
EP-0625143-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1994-11-23 EP disclosed
WO-1993015055-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1993-08-05 WO disclosed