SCHEMBL9128779

SCHEMBL9128779

Cc1ccc(S(=O)(=O)NCCc2cccc(OCCN[C@@H](C)C(=O)O)c2)cc1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
F2 P00734 2/20 0.51
AKR1C3 P42330 4/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
CYP2D6 P10635 1/20 0.48
ALDH1A1 P00352 3/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
RAB9A P51151 1/20 0.46
PLG P00747 1/20 0.46
SGMS1 Q86VZ5 1/20 0.46
TBXA2R P21731 1/20 0.45
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9127737 0.91 F2 (0.62) F2AKR1C3CYP2D6PLGSGMS1
SCHEMBL9129388 0.82 TBXA2R (0.62) AKR1C3L3MBTL1ALDH1A1MEN1KMT2A
SCHEMBL9130159 0.82 DRD4 (0.55) F2L3MBTL1ALDH1A1MEN1KMT2A
SCHEMBL9128548 0.81 ALDH1A1 (0.56) F2AKR1C3L3MBTL1ALDH1A1MEN1
SCHEMBL9129003 0.79 SGMS1 (0.57) AKR1C3ALDH1A1MEN1KMT2ASGMS1
SCHEMBL9129268 0.78 F2 (0.60) F2AKR1C3ALDH1A1PLGSGMS1
SCHEMBL9129275 0.78 F2 (0.60) F2AKR1C3ALDH1A1PLGSGMS1
SCHEMBL3394469 0.77 L3MBTL1 (0.68) AKR1C3L3MBTL1ALDH1A1MEN1KMT2A
SCHEMBL9129394 0.77 SGMS1 (0.74) L3MBTL1ALDH1A1KMT2ARAB9ASGMS1
SCHEMBL9850603 0.77 SGMS1 (0.59) F2AKR1C3PLGSGMS1TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5446065-A Thromboxane antagonists BOEHRINGER MANNHEIM GMBH (DE) 1995-08-29 US disclosed
EP-0564499-B1 NOVEL AMINES, PROCESS FOR PRODUCING THEM AND MEDICAMENTS CONTAINING SAID COMPOUNDS BOEHRINGER MANNHEIM GMBH (DE) 1995-04-12 EP disclosed
EP-0564499-A1 NOVEL AMINES, PROCESS FOR PRODUCING THEM AND MEDICAMENTS CONTAINING SAID COMPOUNDS. BOEHRINGER MANNHEIM GMBH (DE) 1993-10-13 EP disclosed
WO-1992011234-A1 NOVEL AMINES, PROCESS FOR PRODUCING THEM AND MEDICAMENTS CONTAINING SAID COMPOUNDS BOEHRINGER MANNHEIM GMBH (DE) 1992-07-09 WO disclosed