SCHEMBL9130225

SCHEMBL9130225

O=C(Nc1ccccc1OCC1CO1)c1cccc2[nH]ccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
MRGPRX1 Q96LB2 4/20 0.47
DHPS P49366 2/20 0.44
HDAC3 O15379 2/20 0.43
HDAC1 Q13547 2/20 0.43
KDM1A O60341 1/20 0.42
PARP1 P09874 2/20 0.42
HSD17B10 Q99714 1/20 0.42
ALDH1A1 P00352 2/20 0.41
DHFR P00374 1/20 0.41
GLA P06280 1/20 0.40
GFER P55789 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9129615 0.92 DHPS (0.45) NPC1MEN1KMT2AMRGPRX1DHPS
SCHEMBL9450398 0.84 TUBB4A (0.45) NPC1DHPSHDAC3HDAC1ALDH1A1
SCHEMBL9129235 0.84 MEN1 (0.50) NPC1MEN1KMT2AMRGPRX1DHPS
SCHEMBL9795192 0.83 HSD17B10 (0.60) NPC1MEN1KMT2AMRGPRX1DHPS
SCHEMBL9131919 0.83 MEN1 (0.49) NPC1MEN1KMT2AMRGPRX1DHPS
SCHEMBL9795045 0.81 HDAC1 (0.50) NPC1MEN1KMT2AMRGPRX1DHPS
SCHEMBL9132310 0.81 MEN1 (0.50) NPC1MEN1KMT2AMRGPRX1DHPS
SCHEMBL9132467 0.81 DHPS (0.49) DHPSKDM1APARP1
SCHEMBL9795043 0.81 HDAC1 (0.52) NPC1MEN1KMT2AMRGPRX1DHPS
SCHEMBL9133056 0.80 ALDH1A1 (0.44) NPC1MEN1KMT2ADHPSHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5380722-A Antiarrhythmia agents ROUSSEL-UCLAF (FR) 1995-01-10 US disclosed
US-5084455-A Antiarrhythmia agents for mammals ROUSSEL UCLAF (FR) 1992-01-28 US disclosed
US-4908367-A Antiarrythmic agents Uclaf, Roussel (FR) 1990-03-13 US disclosed
US-4791109-A Novel indole carboxamides ROUSSEL UCLAF (FR) 1988-12-13 US disclosed