SCHEMBL9155992

SCHEMBL9155992

CCC1CCC(C(C)c2ccc(-c3ccc(C(F)(F)F)nc3)cc2)CC1

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TRPV3 Q8NET8 5/20 0.40
PTGS2 P35354 1/20 0.40
P2RX7 Q99572 9/20 0.37
PDE2A O00408 3/20 0.35
MCHR1 Q99705 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9152394 0.91 TRPV3 (0.41) TRPV3PTGS2P2RX7
SCHEMBL9161171 0.89 PTGS2 (0.38) TRPV3PTGS2P2RX7PDE2AMCHR1
SCHEMBL9155828 0.88 PTGS2 (0.38) TRPV3PTGS2P2RX7PDE2AMCHR1
SCHEMBL9154581 0.87 PSEN1 (0.38) TRPV3PTGS2P2RX7PDE2AMCHR1
SCHEMBL9158482 0.87 PSEN1 (0.38) TRPV3PTGS2P2RX7PDE2AMCHR1
SCHEMBL9159950 0.87 TRPV3 (0.41) TRPV3P2RX7
SCHEMBL9158975 0.83 PTGS2 (0.37) PTGS2P2RX7
SCHEMBL9158778 0.81 DGAT1 (0.50) TRPV3MCHR1
SCHEMBL9156338 0.81 PIK3CD (0.37)
SCHEMBL9158763 0.81 DGAT1 (0.50) TRPV3MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445248-B1 PYRIDINE DERIVATIVES MERCK PATENT GMBH (DE) 1995-03-08 EP disclosed
WO-1991004248-A1 PYRIDINE DERIVATIVES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1991-04-04 WO disclosed