SCHEMBL9158975

SCHEMBL9158975

CCC1CCC(C(C)c2ccc(-c3ccc(F)nc3)cc2)CC1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.37
GRIA2 P42262 5/20 0.37
KCNH2 Q12809 3/20 0.37
CYP2A6 P11509 3/20 0.35
CYP2B6 P20813 3/20 0.35
CYP2E1 P05181 1/20 0.35
MMP2 P08253 1/20 0.34
MMP9 P14780 1/20 0.34
MMP13 P45452 1/20 0.34
APLNR P35414 2/20 0.34
CYP11B2 P19099 1/20 0.33
AXL P30530 1/20 0.33
TYRO3 Q06418 1/20 0.33
MERTK Q12866 1/20 0.33
P2RX7 Q99572 1/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2C19 P33261 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9766624 0.90 P2RX7 (0.37) P2RX7
SCHEMBL9158474 0.90 PTGS2 (0.36) PTGS2GRIA2KCNH2CYP2A6CYP2B6
SCHEMBL9155759 0.87 PTGS2 (0.35) PTGS2GRIA2KCNH2CYP2A6CYP2B6
SCHEMBL9157491 0.86 PTGS2 (0.35) PTGS2GRIA2KCNH2CYP2A6CYP2B6
SCHEMBL9158940 0.85 GAA (0.35) PTGS2GRIA2KCNH2CYP2A6CYP2B6
SCHEMBL9156816 0.85 GAA (0.35) PTGS2GRIA2KCNH2CYP2A6CYP2B6
SCHEMBL9156338 0.84 PIK3CD (0.37) CYP2A6CYP3A4
SCHEMBL8774169 0.83 GRIN2B (0.36) PTGS2
SCHEMBL9155992 0.83 TRPV3 (0.40) PTGS2P2RX7
SCHEMBL12891848 0.79 SLC6A2 (0.36) GRIA2P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445248-B1 PYRIDINE DERIVATIVES MERCK PATENT GMBH (DE) 1995-03-08 EP disclosed
US-5205962-A Stable liquid crystals MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1993-04-27 US disclosed
WO-1991004248-A1 PYRIDINE DERIVATIVES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1991-04-04 WO disclosed