SCHEMBL9160185

SCHEMBL9160185

COc1ccc(CCN(C)CCCCNC(=O)C/C=C/c2ccc(-c3cc[n+]([O-])cc3)cc2)cc1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.45
TMEM97 Q5BJF2 2/20 0.45
SIGMAR1 Q99720 2/20 0.45
CYP3A4 P08684 4/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
BLM P54132 1/20 0.43
PMP22 Q01453 1/20 0.43
MAPT P10636 6/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
ALDH1A1 P00352 2/20 0.41
OPRK1 P41145 1/20 0.41
OPRD1 P41143 1/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
LMNA P02545 1/20 0.41
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9228273 0.92 OPRM1 (0.41) OPRM1TMEM97SIGMAR1CYP3A4CYP1A2
SCHEMBL8828221 0.86 OPRM1 (0.48) OPRM1TMEM97SIGMAR1CYP3A4CYP1A2
SCHEMBL9162275 0.86 OPRM1 (0.43) OPRM1TMEM97SIGMAR1CYP3A4CYP1A2
SCHEMBL8828131 0.86 CYP3A4 (0.52) OPRM1TMEM97SIGMAR1CYP3A4CYP1A2
SCHEMBL9160110 0.85 PTAFR (0.47) OPRM1TMEM97SIGMAR1CYP3A4CYP1A2
SCHEMBL9231260 0.85 ABCB1 (0.44) OPRM1TMEM97SIGMAR1CYP3A4CYP1A2
SCHEMBL8828235 0.85 MAPT (0.56) OPRM1TMEM97SIGMAR1CYP3A4CYP1A2
SCHEMBL8828147 0.85 MAPT (0.56) OPRM1TMEM97SIGMAR1CYP3A4CYP1A2
SCHEMBL8828188 0.84 LMNA (0.49) OPRM1TMEM97SIGMAR1CYP3A4CYP1A2
SCHEMBL8828274 0.84 OPRM1 (0.49) OPRM1TMEM97SIGMAR1CYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5430059-A Treating heart disease EISAI CO., LTD. (JP) 1995-07-04 US disclosed
EP-0633248-A1 Butenoic acid derivatives Eisai Co., Ltd. (JP) 1995-01-11 EP disclosed
EP-0589491-A1 Butenoic acid derivatives Eisai Co., Ltd. (JP) 1994-03-30 EP disclosed
US-5292770-A Butenoic acid derivatives EISAI CO., LTD. (JP) 1994-03-08 US disclosed
US-5166188-A Cardiovascular disorders, antiischemic agents EISAI CO., LTD. (JP) 1992-11-24 US disclosed
EP-0399358-A2 Butenoic acid derivatives Eisai Co., Ltd. (JP) 1990-11-28 EP disclosed