SCHEMBL9160949

SCHEMBL9160949

COc1ccc(CCN(C)C(C)CCNC(=O)C/C=C/c2ccc(-c3cccnc3)cc2)cc1OC

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.44
SMPD1 P17405 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
MAPT P10636 6/20 0.41
CYP3A4 P08684 3/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
PTAFR P25105 4/20 0.41
ALDH1A1 P00352 2/20 0.40
RXFP1 Q9HBX9 1/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP51A1 Q16850 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8828233 0.87 OPRM1 (0.47) MAPK1SMPD1SMN1; SMN2MAPTCYP3A4
SCHEMBL9160110 0.86 PTAFR (0.47) MAPK1SMPD1SMN1; SMN2MAPTCYP3A4
SCHEMBL8828201 0.83 NOS2 (0.40) MAPTCYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL9235063 0.80 MAPT (0.40) SMN1; SMN2MAPTCYP3A4CYP2C9CYP2C19
SCHEMBL8828139 0.79 ALDH1A1 (0.44) SMPD1PTAFRALDH1A1MEN1KMT2A
SCHEMBL8828221 0.78 OPRM1 (0.48) SMN1; SMN2MAPTCYP3A4CYP2C9CYP2C19
SCHEMBL9282465 0.77 ALDH1A1 (0.39) MAPTCYP3A4CYP2C9CYP2C19CYP2D6
SCHEMBL9159790 0.76 NOS2 (0.39) SMN1; SMN2MAPTALDH1A1MEN1KMT2A
SCHEMBL9044237 0.75 OPRM1 (0.44) MAPK1SMN1; SMN2MAPTCYP3A4CYP2C9
SCHEMBL9160567 0.75 PTAFR (0.46) PTAFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5430059-A Treating heart disease EISAI CO., LTD. (JP) 1995-07-04 US disclosed
EP-0633248-A1 Butenoic acid derivatives Eisai Co., Ltd. (JP) 1995-01-11 EP disclosed
EP-0589491-A1 Butenoic acid derivatives Eisai Co., Ltd. (JP) 1994-03-30 EP disclosed
US-5292770-A Butenoic acid derivatives EISAI CO., LTD. (JP) 1994-03-08 US disclosed
US-5166188-A Cardiovascular disorders, antiischemic agents EISAI CO., LTD. (JP) 1992-11-24 US disclosed