SCHEMBL9182155

SCHEMBL9182155

CCC1=Nc2cc3c(cc2C(=O)C1)OCO3

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.38
ACHE P22303 1/20 0.36
SCN1A P35498 1/20 0.35
SCN2A Q99250 1/20 0.35
SCN3A Q9NY46 1/20 0.35
BRD9 Q9H8M2 2/20 0.35
BRD7 Q9NPI1 1/20 0.35
MAPT P10636 5/20 0.34
MEN1 O00255 4/20 0.34
KMT2A Q03164 4/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
PSMD14 O00487 1/20 0.34
TP53 P04637 1/20 0.34
CASP1 P29466 1/20 0.34
CASP7 P55210 1/20 0.34
KDM4E B2RXH2 4/20 0.33
ALDH1A1 P00352 2/20 0.33
USP2 O75604 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9178830 0.74 KDM4E (0.40) ACHEMAPTMEN1KMT2AKDM4E
SCHEMBL9180722 0.72 KMT2A (0.40) MEN1KMT2AKDM4EALDH1A1HPGD
SCHEMBL9182860 0.71 HPGD (0.36) ACHEMAPTL3MBTL1KDM4EALDH1A1
SCHEMBL20963316 0.70 CYP2D6 (0.47) CYP2D6ACHETDP1KDM4EALDH1A1
SCHEMBL4764684 0.69 SHMT2 (0.39) CYP2D6MAPTMEN1KMT2AL3MBTL1
SCHEMBL9179384 0.69 KDM4E (0.42) KDM4EALDH1A1CYP3A4SMN1; SMN2HTT
SCHEMBL9183312 0.69 PDE3B (0.46) ACHEMAPTKDM4EALDH1A1HPGD
SCHEMBL9180106 0.69 ALDH1A3 (0.32) ALDH1A1TSHR
SCHEMBL9175477 0.69 ALDH1A1 (0.37) TDP1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL18280773 0.68 NPC1 (0.43) ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5444071-A Hypotensive agent IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1995-08-22 US disclosed
EP-0412848-B1 Quinoline derivatives, process for their preparation and their use as medicaments ICI PLC (GB) 1995-01-18 EP disclosed
EP-0412848-A2 Quinoline derivatives, process for their preparation and their use as medicaments ZENECA LIMITED (GB) 1991-02-13 EP disclosed