SCHEMBL918401

SCHEMBL918401

NC(=O)C(N)Cc1ccc(O)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 3/20 0.71
TAAR1 Q96RJ0 3/20 0.55
SLC6A2 P23975 1/20 0.55
HDAC8 Q9BY41 2/20 0.53
CA2 P00918 1/20 0.52
ESR1 P03372 1/20 0.52
ESR2 Q92731 1/20 0.52
PTGS1 P23219 2/20 0.48
ALPI P09923 1/20 0.48
PKM P14618 1/20 0.48
XIAP P98170 1/20 0.48
DPP4 P27487 1/20 0.48
TPH1 P17752 1/20 0.46
KDM4E B2RXH2 1/20 0.46
USP2 O75604 1/20 0.46
EGFR P00533 1/20 0.46
LCK P06239 1/20 0.46
FYN P06241 1/20 0.46
ADORA3 P0DMS8 1/20 0.46
ALOX15 P16050 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL358908 1.00 SLC7A5 (0.71) SLC7A5TAAR1SLC6A2HDAC8CA2
SCHEMBL3241485 1.00 SLC7A5 (0.71) SLC7A5TAAR1SLC6A2HDAC8CA2
Hydrochloric Acid SCHEMBL29401826 0.98 SLC7A5 (0.69) SLC7A5TAAR1SLC6A2HDAC8CA2
Bromide SCHEMBL14832338 0.98 SLC7A5 (0.69) SLC7A5TAAR1SLC6A2HDAC8CA2
Bromide SCHEMBL28349416 0.98 SLC7A5 (0.69) SLC7A5TAAR1SLC6A2HDAC8CA2
Hydrochloric Acid SCHEMBL6693119 0.98 SLC7A5 (0.69) SLC7A5TAAR1SLC6A2HDAC8CA2
Hydrochloric Acid SCHEMBL3166836 0.98 SLC7A5 (0.69) SLC7A5TAAR1SLC6A2HDAC8CA2
Ammonia Solution, Strong SCHEMBL6760516 0.98 SLC7A5 (0.69) SLC7A5TAAR1SLC6A2HDAC8CA2
SCHEMBL5963611 0.98 SLC7A5 (0.69) SLC7A5TAAR1SLC6A2HDAC8CA2
SCHEMBL5792004 0.98 SLC7A5 (0.69) SLC7A5TAAR1SLC6A2HDAC8CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 607 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260027071-A1 COMPOSITION FOR PROMOTING COLLAGEN PRODUCTION COMPRISING AMIDATED AMINO ACID KYUNGPOOK NAT UNIV IND ACADEMIC COOP FOUND (KR) 2026-01-29 US claimed
EP-4680338-A1 METHODS FOR PREPARING APTAMERS FOR SMALL MOLECULES The Trustees Of Columbia University In The City Of New York (US) 2026-01-21 EP claimed
US-20260015619-A1 METHODS FOR PREPARING APTAMERS FOR SMALL MOLECULES UNIV COLUMBIA (US) 2026-01-15 US claimed
EP-4483868-A1 COMPOSITION FOR PROMOTING COLLAGEN PRODUCTION COMPRISING AMIDATED AMINO ACID Boo, Yong Chool (KR) 2025-01-01 EP claimed
WO-2024196785-A1 METHODS FOR PREPARING APTAMERS FOR SMALL MOLECULES THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2024-09-26 WO claimed
CN-118688315-A Multichannel high-coverage synchronous quantification method for amino-containing and hydroxyl-containing compounds 复旦大学 2024-09-24 CN claimed
US-20230363713-A1 HYDROGEL MICRONEEDLES FOR BIOSENSING POUDINEH MAHLA (CA) 2023-11-16 US claimed
WO-2023158164-A1 COMPOSITION FOR PROMOTING COLLAGEN PRODUCTION COMPRISING AMIDATED AMINO ACID 경북대학교 산학협력단 2023-08-24 WO claimed
EP-4045088-A1 METHOD FOR THE PREPARATION OF POLYMERIC CARRIERS FOR PH- CONTROLLED DRUG RELEASE AND THEIR CONJUGATES WITH DRUGS Ustav Makromolekularni Chemie AV CR, v.v.i. (CZ) 2022-08-24 EP claimed
WO-2021073667-A1 METHOD FOR THE PREPARATION OF POLYMERIC CARRIERS FOR PH- CONTROLLED DRUG RELEASE AND THEIR CONJUGATES WITH DRUGS USTAV MAKROMOLEKULARNI CHEMIE AV CR, V.V.I. (CZ) 2021-04-22 WO claimed
WO-1996039165-A1 PEPTIDES AND COMPOUNDS THAT BIND TO THE IL-1 RECEPTOR AFFYMAX TECHNOLOGIES N.V. (GB) 1996-12-12 WO claimed
US-5519000-A OLIGOPEPTIDE CENTECOR, INC. (US) 1996-05-21 US claimed
US-5506340-A POLYPEPTIDE HAVING ACETYLATED AMINO TERMINAL AND/OR AMIDATED CARBOXY TERMINAL CENTECOR, INC. (US) 1996-04-09 US claimed
WO-1995026744-A1 TUMOR NECROSIS FACTOR INHIBITORS CENTOCOR, INC. (US) 1995-10-12 WO claimed
EP-0193113-B1 PROCESS FOR OPTICALLY ISOMERIZING OPTICALLY ACTIVE ALPHA-AMINO ACID AMIDES AND PROCESS FOR PRODUCING OPTICALLY ACTIVE ALPHA-AMINO ACIDS MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) 1992-01-22 EP claimed
US-4918196-A HEATING IN PRESENCE OF STRONG BASE, SOLVENT OR SOLVENT-FREE MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) 1990-04-17 US claimed
US-4725577-A Biologically active lysine containing octapeptides ADMINISTRATORS OF THE TULANE EDUCATIONAL FUND (US) 1988-02-16 US claimed
US-4650787-A SOMATOSTATIN ANALOG ADMINISTRATORS OF THE TULANE EDUCATIONAL FUND OF NEW ORLEANS, LOUISIANA, THE, 1987-03-17 US claimed
EP-0203031-A2 Biologically active lysine containing octapeptides The Administrators of The Tulane University Educational Fund (US) 1986-11-26 EP claimed
EP-0193113-A1 Process for optically isomerizing optically active alpha-amino acid amides and process for producing optically active alpha-amino acids MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) 1986-09-03 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260015619-A1 METHODS FOR PREPARING APTAMERS FOR SMALL MOLECULES HNMT, GNMT, PNMT SLC7A5 307/4885TAAR1 631/4885SLC6A2 68/4885
US-20260027071-A1 COMPOSITION FOR PROMOTING COLLAGEN PRODUCTION COMPRISING AMIDATED AMINO ACID COL2A1, COL14A1, GLS SLC7A5 1146/4885TAAR1 2267/4885SLC6A2 3676/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.