SCHEMBL9185207

SCHEMBL9185207

Cc1ccc(S(=O)(=O)N(CCCNC(=O)OC(C)(C)C)c2ccccc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.50
GAA P10253 1/20 0.50
HTT P42858 1/20 0.50
KEAP1 Q14145 1/20 0.49
NFE2L2 Q16236 1/20 0.49
PTGER1 P34995 1/20 0.48
BMP1 P13497 1/20 0.48
ESR1 P03372 1/20 0.48
MAPT P10636 2/20 0.47
CA12 O43570 4/20 0.47
CA1 P00915 4/20 0.47
CA2 P00918 4/20 0.47
CA9 Q16790 4/20 0.47
KMT2A Q03164 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
TSHR P16473 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
MEN1 O00255 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9186002 0.82 ESR1 (0.50) LMNAGAAHTTKEAP1NFE2L2
SCHEMBL9186195 0.80 ESR1 (0.48) LMNAGAAHTTKEAP1NFE2L2
SCHEMBL9188513 0.80 ESR1 (0.57) LMNAGAAHTTKEAP1NFE2L2
SCHEMBL5704478 0.79 PSEN1 (0.44) LMNAKEAP1NFE2L2MAPTCA12
SCHEMBL9189756 0.78 ESR1 (0.54) LMNAGAAHTTKEAP1NFE2L2
SCHEMBL9186869 0.77 ALOX5 (0.53) LMNAGAAHTTKEAP1NFE2L2
SCHEMBL14502622 0.77 KEAP1 (0.66) LMNAGAAHTTKEAP1NFE2L2
SCHEMBL9100684 0.76 CKS1B (0.52) GAAMAPTCA12CA1CA2
SCHEMBL8466425 0.74 ESR1 (0.76) KEAP1NFE2L2ESR1CA12CA9
SCHEMBL6554383 0.74 CA1 (0.45) GAAKEAP1NFE2L2MAPTCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0497202-B1 Polyamine thiols as radioprotective agents MERRELL DOW PHARMA (US) 1995-09-13 EP disclosed
US-5217964-A POLYAMINE THIOLS AS RADIOPROTECTIVE AGENTS MERRELL DOW PHARMACEUTICALS INC. (US) 1993-06-08 US disclosed
EP-0497202-A1 Polyamine thiols as radioprotective agents MERRELL DOW PHARMACEUTICALS INC. (US) 1992-08-05 EP disclosed