SCHEMBL9186002

SCHEMBL9186002

Cc1ccc(S(=O)(=O)N(CCCN(CCCN(c2ccccc2)S(=O)(=O)c2ccc(C)cc2)C(=O)OC(C)(C)C)c2ccccc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.50
LMNA P02545 2/20 0.49
GAA P10253 1/20 0.49
HTT P42858 1/20 0.49
KEAP1 Q14145 1/20 0.48
NFE2L2 Q16236 1/20 0.48
BMP1 P13497 1/20 0.47
MAPT P10636 1/20 0.47
KMT2A Q03164 3/20 0.47
MEN1 O00255 1/20 0.47
CAMK2A Q9UQM7 2/20 0.45
F2 P00734 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
ALOX5 P09917 1/20 0.45
CAMK2G Q13555 1/20 0.44
HCRTR2 O43614 1/20 0.44
CNR1 P21554 1/20 0.44
CNR2 P34972 1/20 0.44
NR3C1 P04150 1/20 0.44
ALDH1A1 P00352 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9186195 0.98 ESR1 (0.48) ESR1LMNAGAAHTTKEAP1
SCHEMBL9186869 0.94 ALOX5 (0.53) ESR1LMNAGAAHTTKEAP1
SCHEMBL9189262 0.87 ALDH1A1 (0.56) LMNAGAAHTTKEAP1NFE2L2
SCHEMBL9183310 0.83 CNR2 (0.59) HTTBMP1MAPTCNR1CNR2
SCHEMBL9185207 0.82 LMNA (0.50) ESR1LMNAGAAHTTKEAP1
SCHEMBL9189261 0.81 PSEN1 (0.41) KEAP1NFE2L2KMT2AMEN1F2
SCHEMBL8466425 0.76 ESR1 (0.76) ESR1KEAP1NFE2L2KMT2AMEN1
SCHEMBL14502622 0.76 KEAP1 (0.66) ESR1LMNAGAAHTTKEAP1
SCHEMBL9186142 0.75 ESR1 (0.58) ESR1LMNAGAAHTTKEAP1
SCHEMBL6204172 0.75 ESR1 (0.55) ESR1LMNAGAAHTTKEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0497202-B1 Polyamine thiols as radioprotective agents MERRELL DOW PHARMA (US) 1995-09-13 EP disclosed
US-5217964-A POLYAMINE THIOLS AS RADIOPROTECTIVE AGENTS MERRELL DOW PHARMACEUTICALS INC. (US) 1993-06-08 US disclosed
EP-0497202-A1 Polyamine thiols as radioprotective agents MERRELL DOW PHARMACEUTICALS INC. (US) 1992-08-05 EP disclosed