SCHEMBL9192201

SCHEMBL9192201

Cc1cccc(C)c1NC(=O)N(Cc1ccccc1)CC(c1ccccc1)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
NPSR1 Q6W5P4 1/20 0.49
TDP1 Q9NUW8 1/20 0.47
CYP1A2 P05177 2/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
CASR P41180 1/20 0.47
POLB P06746 1/20 0.46
EGFR P00533 2/20 0.46
ERBB2 P04626 2/20 0.46
GAA P10253 1/20 0.45
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
TRPV1 Q8NER1 2/20 0.43
CYP3A4 P08684 1/20 0.42
ALOX12 P18054 1/20 0.42
PTGES O14684 1/20 0.42
LPAR1 Q92633 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11142406 0.87 ALDH1A1 (0.63) ALDH1A1NPSR1TDP1CYP1A2CYP2C9
SCHEMBL9765025 0.85 SOAT2 (0.49) ALDH1A1NPSR1CYP1A2CYP2C9CYP2C19
SCHEMBL9765052 0.80 ICMT (0.46) ALDH1A1NPSR1EGFRMAPK1HDAC1
SCHEMBL11144230 0.78 ALDH1A1 (0.55) ALDH1A1NPSR1TDP1POLBEGFR
SCHEMBL11145395 0.78 ALDH1A1 (0.56) ALDH1A1NPSR1TDP1POLBEGFR
SCHEMBL11134972 0.74 KMT2A (0.51) ALDH1A1CYP1A2CYP2C9CYP2C19GAA
SCHEMBL11137929 0.73 KMT2A (0.64) ALDH1A1NPSR1TDP1POLBEGFR
SCHEMBL9765058 0.73 TP53 (0.46) ALDH1A1NPSR1TDP1CYP2C19POLB
SCHEMBL11139406 0.73 ALDH1A1 (0.63) ALDH1A1NPSR1POLBEGFRERBB2
SCHEMBL30734411 0.73 ALDH1A1 (0.63) ALDH1A1NPSR1POLBEGFRERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0384320-A1 Antihyperlipidemic and anti-atherosclerotic trisubstituted urea compounds WARNER-LAMBERT COMPANY (US) 1990-08-29 EP claimed
EP-0500348-B1 Disubstituted ureas and thioureas PHARMACIA SPA (IT) 1995-05-17 EP disclosed
US-4994465-A Antihyperlipidemic and antiatherosclerotic trisubstituted urea compounds WARNER-LAMBERT COMPANY (US) 1991-02-19 US disclosed
EP-0384320-A1 Antihyperlipidemic and anti-atherosclerotic trisubstituted urea compounds WARNER-LAMBERT COMPANY (US) 1990-08-29 EP disclosed