SCHEMBL9192515

SCHEMBL9192515

CC(=O)N(O)Cc1cccc(C#Cc2cccc3ccccc23)c1

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.48
ACACB O00763 1/20 0.48
PTGES O14684 16/20 0.43
ALOX5 P09917 1/20 0.42
PTGS1 P23219 1/20 0.42
PTGS2 P35354 1/20 0.42
CHAT P28329 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9476552 0.88 HRH3 (0.48) HRH3ACACBPTGESALOX5CHAT
SCHEMBL9192563 0.84 PTGES (0.56) PTGESALOX5PTGS1PTGS2
SCHEMBL9195229 0.84 ACACB (0.48) ACACBPTGESALOX5PTGS1PTGS2
SCHEMBL9193618 0.83 PTGES (0.62) PTGESALOX5PTGS1PTGS2
SCHEMBL9197210 0.77 PTGES (0.58) ACACBPTGESALOX5PTGS1PTGS2
SCHEMBL9299975 0.75 ACACB (0.43) HRH3ACACBALOX5PTGS1PTGS2
SCHEMBL9197316 0.75 PTGES (0.59) ACACBPTGESALOX5PTGS1PTGS2
SCHEMBL9197649 0.75 PTGES (0.59) PTGESALOX5PTGS1PTGS2
SCHEMBL9197154 0.75 PTGES (0.50) ACACBPTGES
SCHEMBL9476517 0.73 FFAR1 (0.41) PTGESALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0468281-B1 Substituted phenylacetylenes, pharmaceuticals containing them and methods for the preparation of these compounds and pharmaceuticals GRUENENTHAL GMBH (DE) 1995-03-08 EP disclosed
US-5202349-A Lipoxygenase inhibitors, antiasthatics GRUENENTHAL GMBH (DE) 1993-04-13 US disclosed
EP-0468281-A1 Substituted phenylacetylenes, pharmaceuticals containing them and methods for the preparation of these compounds and pharmaceuticals Grünenthal GmbH (DE) 1992-01-29 EP disclosed