SCHEMBL9192563

SCHEMBL9192563

CC(=O)N(O)Cc1cccc(C#Cc2ccccc2)c1

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGES O14684 19/20 0.56
ALOX5 P09917 1/20 0.54
PTGS1 P23219 1/20 0.54
PTGS2 P35354 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9197210 0.89 PTGES (0.58) PTGESALOX5PTGS1PTGS2
SCHEMBL9195229 0.88 ACACB (0.48) PTGESALOX5PTGS1PTGS2
SCHEMBL9197154 0.86 PTGES (0.50) PTGES
SCHEMBL9197316 0.86 PTGES (0.59) PTGESALOX5PTGS1PTGS2
SCHEMBL9192515 0.84 HRH3 (0.48) PTGESALOX5PTGS1PTGS2
SCHEMBL9193618 0.84 PTGES (0.62) PTGESALOX5PTGS1PTGS2
SCHEMBL9197649 0.84 PTGES (0.59) PTGESALOX5PTGS1PTGS2
SCHEMBL9300627 0.82 ALOX5 (0.45) PTGESALOX5PTGS1PTGS2
SCHEMBL1436622 0.80 ALOX5 (0.70) ALOX5PTGS1PTGS2
SCHEMBL9707266 0.76 ALOX5 (0.61) PTGESALOX5PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0468281-B1 Substituted phenylacetylenes, pharmaceuticals containing them and methods for the preparation of these compounds and pharmaceuticals GRUENENTHAL GMBH (DE) 1995-03-08 EP disclosed
US-5202349-A Lipoxygenase inhibitors, antiasthatics GRUENENTHAL GMBH (DE) 1993-04-13 US disclosed
EP-0468281-A1 Substituted phenylacetylenes, pharmaceuticals containing them and methods for the preparation of these compounds and pharmaceuticals Grünenthal GmbH (DE) 1992-01-29 EP disclosed