SCHEMBL9197154

SCHEMBL9197154

CC(=O)N(O)Cc1cccc(C#Cc2ccc(C(C)C)cc2)c1

nearest known ligand 0.50

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGES O14684 18/20 0.50
AKR1C3 P42330 3/20 0.47
ACACB O00763 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9197210 0.87 PTGES (0.58) PTGESAKR1C3ACACB
SCHEMBL9192563 0.86 PTGES (0.56) PTGES
SCHEMBL9195229 0.83 ACACB (0.48) PTGESACACB
SCHEMBL9197316 0.82 PTGES (0.59) PTGESACACB
SCHEMBL9192595 0.79 ACACB (0.42) PTGESACACB
SCHEMBL9197649 0.77 PTGES (0.59) PTGESAKR1C3
SCHEMBL9193618 0.75 PTGES (0.62) PTGES
SCHEMBL9192515 0.75 HRH3 (0.48) PTGESACACB
SCHEMBL9300627 0.75 ALOX5 (0.45) PTGES
SCHEMBL9475487 0.74 PTGES (0.55) PTGESAKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0468281-B1 Substituted phenylacetylenes, pharmaceuticals containing them and methods for the preparation of these compounds and pharmaceuticals GRUENENTHAL GMBH (DE) 1995-03-08 EP disclosed
US-5202349-A Lipoxygenase inhibitors, antiasthatics GRUENENTHAL GMBH (DE) 1993-04-13 US disclosed
EP-0468281-A1 Substituted phenylacetylenes, pharmaceuticals containing them and methods for the preparation of these compounds and pharmaceuticals Grünenthal GmbH (DE) 1992-01-29 EP disclosed