SCHEMBL9194197

SCHEMBL9194197

COc1cccc2c1CCNC2=S

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.43
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.42
MAPT P10636 1/20 0.42
ACHE P22303 1/20 0.41
CYP19A1 P11511 2/20 0.41
DCUN1D1 Q96GG9 1/20 0.41
HTR7 P34969 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA4 P22748 1/20 0.40
CA6 P23280 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29688148 0.80 PARP1 (0.63) PARP1ACHECYP19A1
SCHEMBL437787 0.80 PARP1 (0.63) PARP1ACHECYP19A1
SCHEMBL9447443 0.77 PARP1 (0.64) PARP1ACHECYP19A1HTR7
SCHEMBL927341 0.75 HSD11B1 (0.41)
SCHEMBL31158955 0.75 HSD11B1 (0.41)
SCHEMBL15312032 0.72 HTR7 (0.46) HTR7
SCHEMBL6804044 0.72 ACHE (0.46) KDM4ELMNAPOLBMAPTACHE
SCHEMBL6798725 0.69 ABCB1 (0.47) KDM4ELMNAPOLBMAPTACHE
SCHEMBL7269477 0.69 ALDH1A1 (0.54) KDM4EMAPTCYP19A1RAB9A
SCHEMBL9822382 0.69 PARP1 (0.41) PARP1KDM4ELMNAPOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0355750-B1 Substituted dihydroisoquinolinones and related compounds as potentiators of the lethal effects of radiation and certain chemotherapeutic agents; selected compounds, analogs and process WARNER LAMBERT CO (US) 1995-01-25 EP claimed
US-5177075-A Antitumor agents WARNER-LAMBERT COMPANY (US) 1993-01-05 US claimed
US-5177075-A Antitumor agents WARNER-LAMBERT COMPANY (US) 1993-01-05 US disclosed
EP-0355750-A1 Substituted dihydroisoquinolinones and related compounds as potentiators of the lethal effects of radiation and certain chemotherapeutic agents; selected compounds, analogs and process WARNER-LAMBERT COMPANY (US) 1990-02-28 EP disclosed