SCHEMBL9196819

SCHEMBL9196819

CC(C)COc1ccc(C(=O)NC(=N)N)cc1S(C)(=O)=O

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
THRA P10827 1/20 0.40
THRB P10828 1/20 0.40
EP300 Q09472 2/20 0.39
SLC9A1 P19634 2/20 0.38
ALDH1A1 P00352 1/20 0.38
HIF1A Q16665 1/20 0.38
GPR55 Q9Y2T6 1/20 0.38
SCN9A Q15858 4/20 0.37
SCN5A Q14524 3/20 0.37
AAK1 Q2M2I8 1/20 0.37
MYC P01106 2/20 0.37
MAX P61244 2/20 0.37
SLC9A2 Q9UBY0 1/20 0.37
PDE4B Q07343 1/20 0.36
SLC2A1 P11166 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8813862 0.99 THRA (0.40) THRATHRBEP300SLC9A1ALDH1A1
SCHEMBL9189526 0.91 PKM (0.43) EP300ALDH1A1HIF1AGPR55
SCHEMBL9189972 0.83 PKM (0.49) ALDH1A1
SCHEMBL8816709 0.82 SMPD1 (0.52) ALDH1A1
Hydrochloric Acid SCHEMBL8816482 0.82 PKM (0.48) ALDH1A1
Hydrochloric Acid SCHEMBL8814867 0.81 SMPD1 (0.51) ALDH1A1
SCHEMBL8917612 0.81 THRA (0.41) THRATHRBALDH1A1
SCHEMBL8068683 0.80 SMN1; SMN2 (0.41)
SCHEMBL8743820 0.80 SLC9A1 (0.40) SLC9A1ALDH1A1SLC9A2
SCHEMBL9196826 0.79 SLC9A1 (0.62) SLC9A1SLC9A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0416499-B1 Benzoylguanidines, process for their preparation, their use as medicaments as well as medicament containing them HOECHST AG (DE) 1995-04-26 EP disclosed
US-5292755-A USPA benzolyguanidines HOECHST AKTIENGESELLSCHAFT (DE) 1994-03-08 US disclosed
US-5091394-A BENZOYLGUANIDINES, A PROCESS FOR THEIR PREPARATION, THEIR USE AS MEDICAMENTS AND MEDICAMENTS CONTAINING THEM HOECHST AKTIENGESELLSCHAFT (DE) 1992-02-25 US disclosed
EP-0416499-A2 Benzoylguanidines, process for their preparation, their use as medicaments as well as medicament containing them HOECHST AKTIENGESELLSCHAFT (DE) 1991-03-13 EP disclosed