SCHEMBL8917612

SCHEMBL8917612

COCCOCOc1ccc(C(=O)NC(=N)N)cc1S(C)(=O)=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRA P10827 1/20 0.41
THRB P10828 1/20 0.41
MAPT P10636 2/20 0.38
CTNNB1 P35222 1/20 0.37
TP53 P04637 1/20 0.37
RARG P13631 6/20 0.37
RARA P10276 2/20 0.37
RARB P10826 1/20 0.37
F10 P00742 1/20 0.35
LMNA P02545 2/20 0.35
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 2/20 0.35
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8916182 0.84 VCAM1 (0.45) THRATHRBMAPTCTNNB1RARG
SCHEMBL9189972 0.82 PKM (0.49) MAPTF10LMNAALDH1A1MEN1
SCHEMBL8917633 0.81 SLC9A1 (0.51)
Hydrochloric Acid SCHEMBL8816482 0.81 PKM (0.48) MAPTF10LMNAALDH1A1MEN1
SCHEMBL9196819 0.81 THRA (0.40) THRATHRBALDH1A1
Hydrochloric Acid SCHEMBL8813862 0.80 THRA (0.40) THRATHRBMAPTALDH1A1GAA
SCHEMBL8816709 0.79 SMPD1 (0.52) MAPTF10ALDH1A1KDM4EMEN1
Hydrochloric Acid SCHEMBL8814867 0.78 SMPD1 (0.51) MAPTF10ALDH1A1KDM4EMEN1
SCHEMBL8068683 0.77 SMN1; SMN2 (0.41) MAPTF10LMNAKDM4E
Hydrochloric Acid SCHEMBL8059609 0.76 SMN1; SMN2 (0.40) MAPTF10LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5670544-A ANTIISCHEMIC AGENTS HOECHST AKTIENGESELLSCHAFT (DE) 1997-09-23 US disclosed
EP-0602522-B1 Substituted Benzoylguanidines, method for their preparation, their use as antiarrhythmic agents HOECHST AG (DE) 1996-05-29 EP disclosed
EP-0602522-A1 Substituted Benzoylguanidines, method for their preparation, their use as antiarrhythmic agents HOECHST AKTIENGESELLSCHAFT (DE) 1994-06-22 EP disclosed