SCHEMBL9197878

SCHEMBL9197878

CCn1cccc(C2c3cc(Br)ccc3OC(C)(C)C2O)c1=O

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 8/20 0.37
KCNE1 P15382 7/20 0.37
KCNQ1 P51787 7/20 0.37
NPSR1 Q6W5P4 1/20 0.34
KCNA5 P22460 1/20 0.34
SLC10A2 Q12908 1/20 0.33
MEN1 O00255 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
KCND3 Q9UK17 1/20 0.33
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9199615 0.89 ABCB1 (0.39) ABCC9KCNE1KCNQ1NPSR1CYP3A4
SCHEMBL9199563 0.86 ABCC9 (0.38) ABCC9KCNE1KCNQ1CYP1A2CYP2D6
SCHEMBL9197589 0.84 MAPT (0.43) ABCC9MEN1KMT2A
SCHEMBL9195596 0.84 ABCC9 (0.52) ABCC9KCNE1KCNQ1MEN1CYP1A2
SCHEMBL9197886 0.84 ABCC9 (0.42) ABCC9KCNE1KCNQ1NPSR1MEN1
SCHEMBL9192434 0.82 KCNA5 (0.39) ABCC9KCNA5
SCHEMBL9195248 0.77 SMN1; SMN2 (0.43) KCNE1KCNQ1NPSR1MEN1KMT2A
SCHEMBL9194242 0.77 TP53 (0.46) ABCC9KCNE1KCNQ1NPSR1MEN1
SCHEMBL9682025 0.76 LMNA (0.34) ABCC9KCNE1KCNQ1KCNA5
SCHEMBL9195978 0.74 ABCB1 (0.56) ABCC9CYP1A2CYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0406656-B1 Chroman derivatives MERCK PATENT GMBH (DE) 1995-01-11 EP disclosed
US-5112839-A CHROMAN DERIVATIVES MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-05-12 US disclosed
EP-0406656-A1 Chroman derivatives MERCK PATENT GmbH (DE) 1991-01-09 EP disclosed