SCHEMBL9200327

SCHEMBL9200327

CCOc1ccc2oc(C(CN)CC(=O)O)cc2c1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
HPGD P15428 3/20 0.45
HSD17B10 Q99714 2/20 0.45
MEN1 O00255 1/20 0.45
POLB P06746 1/20 0.45
BLM P54132 1/20 0.45
KMT2A Q03164 1/20 0.45
KDM4E B2RXH2 3/20 0.43
AKR1C3 P42330 1/20 0.43
AKR1C2 P52895 1/20 0.43
TAS1R3 Q7RTX0 3/20 0.40
TAS1R1 Q7RTX1 3/20 0.40
MAPK1 P28482 1/20 0.40
RECQL P46063 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CYP1A2 P05177 1/20 0.40
CA4 P22748 1/20 0.40
CA6 P23280 1/20 0.40
CA5A P35218 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9203506 0.81 LMNA (0.43) MEN1BLMKMT2AAKR1C3AKR1C2
SCHEMBL9196674 0.81 MAOB (0.47) MEN1BLMKMT2ATAS1R3TAS1R1
SCHEMBL9315754 0.79 PIM1 (0.55) ALDH1A1MAPK1CA12CA1CA9
SCHEMBL9198993 0.79 GABBR2 (0.44) MEN1BLMKMT2AKDM4ECYP1A2
SCHEMBL9202393 0.78 GABBR2 (0.54) ALDH1A1HSD17B10MEN1BLMKMT2A
SCHEMBL9196666 0.78 GABBR2 (0.43) MEN1BLMKMT2ACA12CA1
SCHEMBL9315720 0.78 AKR1C3 (0.46) ALDH1A1HPGDHSD17B10MEN1POLB
SCHEMBL9195312 0.78 GAA (0.43) ALDH1A1MEN1BLMKMT2ACYP1A2
SCHEMBL9200322 0.76 AKR1C3 (0.41) ALDH1A1HPGDHSD17B10MEN1POLB
SCHEMBL5866928 0.76 ALDH1A1 (0.68) ALDH1A1HPGDHSD17B10MEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0463969-B1 New compounds of 4-aminobutyric acid, process for their preparation and pharmaceutical preparations containing them ADIR (FR) 1995-02-08 EP claimed
US-5162364-A Treatment of spastic and senescence disorders ADIR ET COMPAGNIE (FR) 1992-11-10 US disclosed