SCHEMBL9201233

SCHEMBL9201233

CCCC(c1ccncc1)n1ccc2cc(C)ccc21

nearest known ligand 0.70

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 8/20 0.70
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
SLC6A4 P31645 4/20 0.39
CYP17A1 P05093 1/20 0.38
ROCK1 Q13464 1/20 0.36
BRD4 O60885 1/20 0.35
ITGB3 P05106 1/20 0.35
ITGAV P06756 1/20 0.35
CYP19A1 P11511 2/20 0.33
SMO Q99835 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8845768 0.86 SLC6A2 (0.68) SLC6A2SLC6A4CYP17A1ITGB3ITGAV
SCHEMBL9197969 0.84 SLC6A2 (0.65) SLC6A2HTR2CSLC6A4CYP17A1ROCK1
SCHEMBL9195174 0.82 SLC6A2 (1.00) SLC6A2SLC6A4CYP17A1
SCHEMBL9192640 0.80 SLC6A2 (0.57) SLC6A2ITGB3ITGAVSMO
SCHEMBL8845698 0.78 SLC6A2 (0.68) SLC6A2SLC6A4CYP17A1
SCHEMBL9194455 0.77 SLC6A2 (0.63) SLC6A2SLC6A4ROCK1ITGB3ITGAV
SCHEMBL9198601 0.77 SLC6A2 (0.59) SLC6A2SLC6A4CYP17A1ITGB3ITGAV
SCHEMBL9155328 0.77 SLC6A2 (0.56) SLC6A2ITGB3ITGAV
SCHEMBL8845539 0.77 SLC6A2 (0.56) SLC6A2SLC6A4ITGB3ITGAV
SCHEMBL15024791 0.76 BRD4 (0.51) SLC6A2HTR2AHTR2CSLC6A4ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0471296-B1 1-(Pyridinylalkyl)-1H-indoles, indolines and related analogs HOECHST ROUSSEL PHARMA (US) 1995-11-08 EP disclosed
US-5214058-A Acetylcholinesterase inhibitors, treatment of senile dementia HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1993-05-25 US disclosed
EP-0471296-A1 1-(Pyridinylalkyl)-1H-indoles, indolines and related analogs HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-02-19 EP disclosed