SCHEMBL9204902

SCHEMBL9204902

COc1cc2c(cc1OC)CC(=O)N(CC1CCCCNC1)CC2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.47
GAA P10253 1/20 0.47
HCN4 Q9Y3Q4 3/20 0.44
CHRM2 P08172 1/20 0.44
HTR1A P08908 1/20 0.44
SLC6A4 P31645 1/20 0.44
DRD3 P35462 1/20 0.44
KCNH2 Q12809 1/20 0.44
MAPT P10636 1/20 0.42
CYP3A4 P08684 1/20 0.42
ALOX15 P16050 1/20 0.42
RAB9A P51151 1/20 0.39
DRD2 P14416 1/20 0.39
ACHE P22303 1/20 0.38
HTR2C P28335 2/20 0.38
HTR2B P41595 1/20 0.38
EHMT2 Q96KQ7 2/20 0.37
ROCK2 O75116 1/20 0.37
KLK7 P49862 1/20 0.36
MDM4 O15151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9212186 0.97 SMN1; SMN2 (0.48) SMN1; SMN2GAAHCN4CHRM2HTR1A
SCHEMBL9215737 0.88 DRD2 (0.40) HCN4CHRM2HTR1ASLC6A4DRD3
SCHEMBL9208378 0.87 MEN1 (0.47) ALOX15DRD2ACHEHTR2CHTR2B
SCHEMBL9216770 0.86 MEN1 (0.46) ALOX15DRD2ACHEHTR2CHTR2B
SCHEMBL9216049 0.83 MEN1 (0.48) HTR1ADRD3DRD2ACHEHTR2C
SCHEMBL9207567 0.83 DRD2 (0.39) SMN1; SMN2DRD2
SCHEMBL9740805 0.81 PARP1 (0.45) DRD2ACHEHTR2CHTR2B
SCHEMBL9739351 0.79 ITGB3 (0.36) SMN1; SMN2GAAHCN4CHRM2HTR1A
SCHEMBL9740567 0.79 DRD2 (0.41) KCNH2DRD2
SCHEMBL9209711 0.79 MEN1 (0.50) SMN1; SMN2MAPTHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0224794-B1 CYCLIC AMINE DERIVATIVES, MEDICINES CONTAINING THESE COMPOUNDS AND PROCESS FOR THEIR PREPARATION Dr. Karl Thomae GmbH (DE) 1990-09-12 EP disclosed
EP-0224794-A2 Cyclic amine derivatives, medicines containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1987-06-10 EP disclosed