SCHEMBL9215737

SCHEMBL9215737

Cc1cc2c(cc1C)CC(=O)N(CC1CCCCNC1)CC2

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.40
PARP1 P09874 1/20 0.37
BRD4 O60885 3/20 0.35
GRM5 P41594 1/20 0.34
KHK P50053 1/20 0.34
CDK9 P50750 1/20 0.33
SYK P43405 1/20 0.33
NAAA Q02083 1/20 0.33
GNRHR P30968 1/20 0.33
ATAD2 Q6PL18 1/20 0.32
KCNH2 Q12809 3/20 0.32
CCR2 P41597 1/20 0.32
GHSR Q92847 1/20 0.32
CHRM2 P08172 1/20 0.31
HTR1A P08908 1/20 0.31
SLC6A4 P31645 1/20 0.31
DRD3 P35462 1/20 0.31
HCN4 Q9Y3Q4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9739351 0.92 ITGB3 (0.36) DRD2PARP1BRD4GRM5KHK
SCHEMBL9204902 0.88 SMN1; SMN2 (0.47) DRD2KCNH2CHRM2HTR1ASLC6A4
SCHEMBL9214240 0.86 GRM5 (0.43) DRD2PARP1BRD4GRM5KHK
SCHEMBL9207567 0.85 DRD2 (0.39) DRD2PARP1GRM5CDK9NAAA
SCHEMBL9212186 0.84 SMN1; SMN2 (0.48) DRD2PARP1KCNH2CHRM2HTR1A
SCHEMBL9740805 0.83 PARP1 (0.45) DRD2PARP1GRM5KHK
SCHEMBL9208151 0.82 GRM5 (0.44) DRD2PARP1BRD4GRM5KHK
SCHEMBL9740567 0.82 DRD2 (0.41) DRD2PARP1GRM5KHKCDK9
SCHEMBL9740563 0.78 DRD2 (0.39) DRD2PARP1GRM5KHKCDK9
SCHEMBL9208356 0.77 GRM5 (0.42) DRD2PARP1GRM5KHKCDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed