SCHEMBL9205290

SCHEMBL9205290

COc1ccc2cc(OCCCCl)ccc2c1OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 7/20 0.47
IDO1 P14902 6/20 0.47
TUBB4A P04350 3/20 0.41
TUBB P07437 3/20 0.41
TUBA3C P0DPH7 3/20 0.41
TUBA1B P68363 3/20 0.41
TUBA4A P68366 3/20 0.41
TUBB4B P68371 3/20 0.41
TUBB3 Q13509 3/20 0.41
TUBB2A Q13885 3/20 0.41
TUBB8 Q3ZCM7 3/20 0.41
TUBA3E Q6PEY2 3/20 0.41
TUBA1A Q71U36 3/20 0.41
TUBA1C Q9BQE3 3/20 0.41
TUBB6 Q9BUF5 3/20 0.41
TUBB2B Q9BVA1 3/20 0.41
TUBB1 Q9H4B7 3/20 0.41
MAPK1 P28482 1/20 0.41
MAPT P10636 2/20 0.40
CYP3A4 P08684 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19612326 0.84 CNR2 (0.46) TDO2IDO1TUBB4ATUBBTUBA3C
SCHEMBL50546 0.81 IDO1 (0.56) TDO2IDO1TUBB4ATUBBTUBA3C
SCHEMBL19612468 0.80 THRA (0.44) MAPK1
SCHEMBL9213813 0.79 PPARG (0.55) MAPK1CYP3A4PPARGALDH1A1
SCHEMBL9211531 0.77 CA2 (0.57) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL19612353 0.77 TUBB1 (0.48) TDO2IDO1TUBB4ATUBBTUBA3C
SCHEMBL9740557 0.76 PPARG (0.56) MAPK1CYP3A4PPARGALDH1A1L3MBTL1
SCHEMBL670196 0.75 MAPK1 (0.45) MAPK1MAPTPPARGKCNA3SLC6A2
SCHEMBL31648415 0.74 L3MBTL1 (0.46) TUBB1MAPK1MAPTALDH1A1LMNA
SCHEMBL6085554 0.73 TDP1 (0.55) MAPK1MAPTPPARGHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed