SCHEMBL9206799

SCHEMBL9206799

O=C(O)CN1CCN(CC(=O)O)Cc2cc(N3CCCC3)cc(n2)CN(CC(=O)O)CC1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 2/20 0.39
ALDH1A1 P00352 3/20 0.38
MAPT P10636 3/20 0.38
KDM4E B2RXH2 1/20 0.38
POLB P06746 1/20 0.38
GAA P10253 1/20 0.38
RAD52 P43351 1/20 0.38
JAK2 O60674 1/20 0.37
SYK P43405 1/20 0.37
MEN1 O00255 1/20 0.37
TSHR P16473 1/20 0.37
KMT2A Q03164 1/20 0.37
GFER P55789 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
S1PR3 Q99500 1/20 0.36
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
GRK6 P43250 1/20 0.36
SLC27A1 Q6PCB7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9207391 0.87 HSD17B10 (0.49) S1PR1ALDH1A1MAPTPOLBMEN1
SCHEMBL9210619 0.80 GABRA1 (0.36) ALDH1A1MAPTKDM4EMEN1TSHR
SCHEMBL9212767 0.80 SLC6A9 (0.47) ALDH1A1MAPTITGB3ITGA2B
SCHEMBL5551311 0.80 SLC6A9 (0.37) S1PR1ITGB3ITGA2B
SCHEMBL9288210 0.79 SLC6A9 (0.36) S1PR1ALDH1A1GAAITGB3ITGA2B
SCHEMBL9288230 0.79 SLC6A9 (0.36) S1PR1ALDH1A1GAAITGB3ITGA2B
SCHEMBL9273384 0.77 SLC6A9 (0.35) S1PR1ALDH1A1MAPTKDM4EITGB3
SCHEMBL9273370 0.77 KCNA5 (0.36) ALDH1A1KDM4EJAK2SYKITGB3
SCHEMBL9206903 0.77 ALDH1A1 (0.43) ALDH1A1MAPTKDM4EMEN1KMT2A
SCHEMBL1394889 0.76 SLC6A9 (0.42) ALDH1A1MAPTPOLBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5403572-A Macrocyclic polyaza compounds containing 5 or 6 membered rings, process for producing them and pharmaceutical media containing them SCHERING AKTIENGESELLSCHAFT (DE) 1995-04-04 US disclosed
EP-0352218-B1 Macrocyclic polyaza compounds containing rings with 5 or 6 members, methods for their preparation and pharmaceutical compositions containing same SCHERING AG (DE) 1995-02-22 EP disclosed
US-5334371-A Marcocyclic polyaza bicyclo compounds containing 5 or 6 membered rings, and method for MRI SCHERING AKTIENGESELLSCHAFT (DE) 1994-08-02 US disclosed
EP-0352218-A2 Macrocyclic polyaza compounds containing rings with 5 or 6 members, methods for their preparation and pharmaceutical compositions containing same SCHERING AKTIENGESELLSCHAFT (DE) 1990-01-24 EP disclosed