SCHEMBL9212767

SCHEMBL9212767

O=C(O)CN1CCN(CC(=O)O)Cc2cc(Cl)cc(n2)CN(CC(=O)O)CC1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 1/20 0.47
CXCR4 P61073 2/20 0.40
MAPK11 Q15759 1/20 0.38
MAPK14 Q16539 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
KMO O15229 1/20 0.37
HSD17B10 Q99714 1/20 0.37
ALDH1A1 P00352 2/20 0.37
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
ITGB3 P05106 1/20 0.35
ITGA2B P08514 1/20 0.35
ATM Q13315 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5551311 0.84 SLC6A9 (0.37) SLC6A9HSD17B10DRD2ITGB3ITGA2B
SCHEMBL9288230 0.83 SLC6A9 (0.36) SLC6A9HSD17B10ALDH1A1ITGB3ITGA2B
SCHEMBL9288210 0.83 SLC6A9 (0.36) SLC6A9HSD17B10ALDH1A1ITGB3ITGA2B
SCHEMBL9206903 0.80 ALDH1A1 (0.43) ALDH1A1LMNAMAPT
SCHEMBL9273384 0.80 SLC6A9 (0.35) SLC6A9HSD17B10ALDH1A1MAPTITGB3
SCHEMBL9206799 0.80 S1PR1 (0.39) ALDH1A1MAPTITGB3ITGA2B
SCHEMBL9273370 0.80 KCNA5 (0.36) SLC6A9HSD17B10ALDH1A1ITGB3ITGA2B
SCHEMBL1394889 0.80 SLC6A9 (0.42) SLC6A9HSD17B10ALDH1A1MAPT
SCHEMBL5556103 0.79 ALDH1A1 (0.38) CXCR4ALDH1A1DRD2
SCHEMBL9205301 0.78 EGLN1 (0.40) SLC6A9HSD17B10ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5403572-A Macrocyclic polyaza compounds containing 5 or 6 membered rings, process for producing them and pharmaceutical media containing them SCHERING AKTIENGESELLSCHAFT (DE) 1995-04-04 US disclosed
EP-0352218-B1 Macrocyclic polyaza compounds containing rings with 5 or 6 members, methods for their preparation and pharmaceutical compositions containing same SCHERING AG (DE) 1995-02-22 EP disclosed
US-5334371-A Marcocyclic polyaza bicyclo compounds containing 5 or 6 membered rings, and method for MRI SCHERING AKTIENGESELLSCHAFT (DE) 1994-08-02 US disclosed
EP-0352218-A2 Macrocyclic polyaza compounds containing rings with 5 or 6 members, methods for their preparation and pharmaceutical compositions containing same SCHERING AKTIENGESELLSCHAFT (DE) 1990-01-24 EP disclosed