SCHEMBL9273370

SCHEMBL9273370

O=C(O)CN1CCN(CC(=O)O)Cc2cc(OCCOc3cc4nc(c3)CN(CC(=O)O)CCN(CC(=O)O)CCN(CC(=O)O)C4)cc(n2)CN(CC(=O)O)CC1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 5/20 0.36
SCN9A Q15858 1/20 0.35
SLC6A9 P48067 1/20 0.35
ITGB3 P05106 1/20 0.34
ITGA2B P08514 1/20 0.34
HSD17B10 Q99714 1/20 0.34
JAK2 O60674 1/20 0.33
SYK P43405 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9206903 0.85 ALDH1A1 (0.43) KDM4EALDH1A1
SCHEMBL5551311 0.80 SLC6A9 (0.37) SCN9ASLC6A9ITGB3ITGA2BHSD17B10
SCHEMBL9212767 0.80 SLC6A9 (0.47) SLC6A9ITGB3ITGA2BHSD17B10ALDH1A1
SCHEMBL9288230 0.79 SLC6A9 (0.36) SCN9ASLC6A9ITGB3ITGA2BHSD17B10
SCHEMBL9288210 0.79 SLC6A9 (0.36) SCN9ASLC6A9ITGB3ITGA2BHSD17B10
SCHEMBL9206799 0.77 S1PR1 (0.39) ITGB3ITGA2BJAK2SYKKDM4E
SCHEMBL9273384 0.77 SLC6A9 (0.35) SCN9ASLC6A9ITGB3ITGA2BHSD17B10
SCHEMBL1394889 0.76 SLC6A9 (0.42) SLC6A9HSD17B10ALDH1A1
SCHEMBL18915193 0.75 ADRB1 (0.40)
SCHEMBL9205301 0.74 EGLN1 (0.40) SLC6A9HSD17B10KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5403572-A Macrocyclic polyaza compounds containing 5 or 6 membered rings, process for producing them and pharmaceutical media containing them SCHERING AKTIENGESELLSCHAFT (DE) 1995-04-04 US disclosed
US-5334371-A Marcocyclic polyaza bicyclo compounds containing 5 or 6 membered rings, and method for MRI SCHERING AKTIENGESELLSCHAFT (DE) 1994-08-02 US disclosed