SCHEMBL9207494

SCHEMBL9207494

COc1cc2c(cc1OC)C(=O)N(CC1CCCNC1)C2

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.48
DRD2 P14416 1/20 0.40
ACHE P22303 1/20 0.40
HTR2A P28223 4/20 0.39
EED O75530 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HTR2C P28335 3/20 0.38
HTR2B P41595 1/20 0.38
EHMT2 Q96KQ7 2/20 0.37
ROCK2 O75116 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9216049 0.89 MEN1 (0.48) PARP1DRD2ACHEHTR2AMEN1
SCHEMBL9208378 0.85 MEN1 (0.47) DRD2ACHEHTR2AMEN1KMT2A
SCHEMBL9216770 0.84 MEN1 (0.46) DRD2ACHEHTR2AMEN1KMT2A
SCHEMBL9209711 0.81 MEN1 (0.50) HTR2AMEN1KMT2AHTR2CHTR2B
SCHEMBL9204844 0.80 MEN1 (0.49) ACHEHTR2AMEN1KMT2AHTR2C
SCHEMBL9212186 0.80 SMN1; SMN2 (0.48) PARP1DRD2HTR2AEEDHTR2C
SCHEMBL9216697 0.79 EED (0.44) ACHEHTR2AEEDHTR2CHTR2B
SCHEMBL9207673 0.78 MEN1 (0.47) DRD2MEN1KMT2A
SCHEMBL9204902 0.76 SMN1; SMN2 (0.47) DRD2ACHEHTR2CHTR2BEHMT2
SCHEMBL16858398 0.76 ACHE (0.43) ACHEHTR2AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed