SCHEMBL9210352

SCHEMBL9210352

COc1ccc(Oc2[nH]c3ccccc3c2CCN)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 3/20 0.50
HTR1D P28221 1/20 0.50
MTNR1A P48039 1/20 0.49
MTNR1B P49286 1/20 0.49
KDM4E B2RXH2 4/20 0.49
KMT2A Q03164 4/20 0.49
MAPT P10636 2/20 0.49
MEN1 O00255 3/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 2/20 0.44
HSD17B10 Q99714 1/20 0.44
TAAR1 Q96RJ0 1/20 0.42
PTGS1 P23219 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TRPM8 Q7Z2W7 1/20 0.41
ABCG2 Q9UNQ0 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29128851 0.85 HTR6 (0.52) HTR6HTR1DKDM4EKMT2AMAPT
SCHEMBL7613059 0.82 KDM4E (0.64) HTR6HTR1DMTNR1AMTNR1BKDM4E
SCHEMBL16299526 0.74 CYP19A1 (0.53) HTR6HTR1DMTNR1AMTNR1BKDM4E
SCHEMBL8508265 0.73 KDM4E (0.56) HTR6HTR1DKDM4EKMT2AMAPT
SCHEMBL1424220 0.71 ALDH1A1 (0.69) HTR6HTR1DKDM4EMAPTALDH1A1
SCHEMBL29415611 0.71 ALDH1A1 (0.69) HTR6HTR1DKDM4EMAPTALDH1A1
Hydrochloric Acid SCHEMBL7401442 0.70 LTA4H (0.55) HTR6HTR1DKDM4EMAPTTRPM8
SCHEMBL8947088 0.70 HTR6 (0.73) HTR6HTR1DMTNR1AMTNR1BKDM4E
SCHEMBL9300309 0.70 HTR6 (0.49) HTR6HTR1DMTNR1AMTNR1BKDM4E
Hydrochloric Acid SCHEMBL273338 0.69 ALDH1A1 (0.67) HTR6HTR1DKDM4EMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0674619-A1 TRYPTAMINE ANALOGUES AS 5-HT 1?-LIKE AGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-10-04 EP disclosed
WO-1994014770-A1 TRYPTAMINE ANALOGUES AS 5-HT1-LIKE AGONISTS SMITHKLINE BEECHAM PLC (GB) 1994-07-07 WO disclosed