SCHEMBL8947088

SCHEMBL8947088

COc1ccc2[nH]c(-c3ccccc3)c(CCN)c2c1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 4/20 0.73
HTR1D P28221 2/20 0.73
HTR1A P08908 1/20 0.73
SLC6A4 P31645 1/20 0.73
HTR7 P34969 1/20 0.73
HTR5A P47898 1/20 0.73
MTNR1A P48039 4/20 0.66
MTNR1B P49286 4/20 0.66
KDM4E B2RXH2 2/20 0.66
ALDH1A1 P00352 1/20 0.66
CYP1A2 P05177 1/20 0.66
CYP3A4 P08684 1/20 0.66
CYP2D6 P10635 1/20 0.66
CYP2C9 P11712 1/20 0.66
HPGD P15428 1/20 0.66
CYP2C19 P33261 1/20 0.66
HSD17B10 Q99714 1/20 0.66
TUBB4A P04350 1/20 0.62
TUBB P07437 1/20 0.62
TUBA3C P0DPH7 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7613059 0.85 KDM4E (0.64) HTR6HTR1DHTR1ASLC6A4HTR7
SCHEMBL29423321 0.85 HTR6 (1.00) HTR6HTR1DHTR1ASLC6A4HTR7
SCHEMBL5763578 0.85 HTR6 (1.00) HTR6HTR1DHTR1ASLC6A4HTR7
SCHEMBL8946961 0.81 HTR6 (0.72) HTR6HTR1DHTR1ASLC6A4HTR7
Oxalic Acid SCHEMBL5781188 0.80 HTR6 (0.89) HTR6HTR1DHTR1ASLC6A4HTR7
SCHEMBL3508630 0.80 MTNR1A (1.00) MTNR1AMTNR1BKDM4EALDH1A1CYP1A2
SCHEMBL29759426 0.80 MTNR1A (1.00) MTNR1AMTNR1BKDM4EALDH1A1CYP1A2
SCHEMBL4875370 0.80 HTR6 (0.70) HTR6KDM4EALDH1A1MAPTKMT2A
SCHEMBL8802574 0.80 MTNR1A (0.67) HTR6HTR1DHTR1ASLC6A4HTR7
SCHEMBL4244966 0.79 HTR1D (1.00) HTR6HTR1DHTR1AHTR7HTR5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5552428-A ANTIARRHYTHMIA AGENTS FOR CARDIOVASCULAR DISORDERS USING MELATONIN DERIVATIVES INSTITUTO FARMACOLOGICO LOMBARDO-IFLO, S.A.S. (IT) 1996-09-03 US disclosed