Bromide

Bromide

SCHEMBL9210496

Br.CC[C@H](C(=O)OC)[C@H](N)C(=O)O

nearest known ligand 0.42

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 1/20 0.33
CHRM3 known ✓ P20309 1/20 0.32
ADRA1A known ✓ P35348 1/20 0.32
SLC6A3 known ✓ Q01959 1/20 0.32
SLC1A1 P43005 5/20 0.42
SLC1A3 P43003 4/20 0.42
SLC1A2 P43004 4/20 0.42
SLC7A5 Q01650 1/20 0.38
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
GLO1 Q04760 1/20 0.37
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CHRM1 P11229 1/20 0.32
AKR1A1 P14550 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HRH1 P35367 1/20 0.32
DRD3 P35462 1/20 0.32
HDAC1 Q13547 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL9213394 0.84 ALOX15 (0.38) SLC1A1SLC1A3SLC1A2SLC7A5GLO1
Bromide SCHEMBL9295134 0.82 CA2 (0.49) SLC1A1SLC1A3SLC1A2CA1CA2
Bromide SCHEMBL9295139 0.82 CA2 (0.49) SLC1A1SLC1A3SLC1A2CA1CA2
SCHEMBL9203696 0.79 CA2 (0.50) SLC1A1SLC1A3SLC1A2CA1CA2
SCHEMBL4753756 0.79 CA1 (0.42) CA1CA2MEN1KMT2ACHRM1
SCHEMBL4753760 0.79 CA1 (0.42) CA1CA2MEN1KMT2ACHRM1
SCHEMBL15015843 0.79 CA1 (0.42) CA1CA2MEN1KMT2ACHRM1
SCHEMBL8982021 0.78 GLO1 (0.48) SLC1A1SLC1A3SLC1A2SLC7A5GLO1
SCHEMBL4902637 0.78 GLO1 (0.48) SLC1A1SLC1A3SLC1A2SLC7A5GLO1
SCHEMBL19525723 0.78 GLO1 (0.48) SLC1A1SLC1A3SLC1A2SLC7A5GLO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0643710-A1 SYNTHESIS OF OPTICALLY ACTIVE LACTONES FROM L-ASPARTIC ACID AND INTERMEDIATES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-03-22 EP disclosed
US-5322942-A Deprotecting and hydrolyzing protected aspartic acid diester, reacting with nitrosylating agent in presence of hydrogen halide, esterifying, reacting with acyl aryl derivative REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1994-06-21 US disclosed
WO-1992021675-A1 SYNTHESIS OF OPTICALLY ACTIVE LACTONES FROM L-ASPARTIC ACID AND INTERMEDIATES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1992-12-10 WO disclosed