SCHEMBL9211

SCHEMBL9211

CCOC(=O)C(C)(C)c1ccc(Br)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
LMNA P02545 2/20 0.49
NPSR1 Q6W5P4 2/20 0.49
CYP1A2 P05177 2/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
CNR2 P34972 7/20 0.48
RORC P51449 1/20 0.47
MAPT P10636 2/20 0.46
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
S1PR4 O95977 1/20 0.46
S1PR1 P21453 1/20 0.46
MAPK1 P28482 1/20 0.46
MMP8 P22894 1/20 0.42
HTT P42858 1/20 0.42
ABCB11 O95342 1/20 0.41
CYP3A4 P08684 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12002476 0.95 CNR2 (0.48) ALDH1A1LMNANPSR1CYP1A2CYP2C9
Tetrahydrofuran SCHEMBL28259594 0.88 ALDH1A1 (0.41) ALDH1A1LMNANPSR1CYP1A2CYP2C9
SCHEMBL18982867 0.86 ALDH1A1 (0.49) ALDH1A1LMNANPSR1CYP1A2CYP2C9
SCHEMBL1684350 0.86 ALDH1A1 (0.49) ALDH1A1LMNANPSR1CYP1A2CYP2C9
SCHEMBL6279399 0.85 CNR2 (0.58) NPSR1CYP1A2SMN1; SMN2CNR2RORC
SCHEMBL23291809 0.84 ALDH1A1 (0.48) ALDH1A1LMNANPSR1CYP1A2CYP2C9
SCHEMBL27568527 0.84 CNR2 (0.47) LMNANPSR1CYP1A2CNR2RORC
SCHEMBL4115523 0.84 CNR2 (0.53) ALDH1A1LMNACNR2RORCKMT2A
SCHEMBL11384534 0.84 ALDH1A1 (0.50) ALDH1A1LMNANPSR1CYP1A2CYP2C9
SCHEMBL6135621 0.83 NPSR1 (0.50) ALDH1A1LMNANPSR1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 141 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12527776-B2 Treatment of ciliopathies using inhibitors of glucosylceramide synthase (GCS) GENZYME CORPORATION (US) 2026-01-20 US disclosed
EP-3920912-B1 TREATMENT OF CILIOPATHIES USING INHIBITORS OF GLUCOSYLCERAMIDE SYNTHASE (GCS) GENZYME CORP (US) 2025-06-11 EP disclosed
US-20250026749-A1 GLUCOSYLCERAMIDE SYNTHASE INHIBITORS GENZYME CORPORATION (US) 2025-01-23 US disclosed
US-12083115-B2 Methods for treating neurological symptoms associated with lysosomal storage diseases GENZYME CORPORATION (US) 2024-09-10 US disclosed
US-12060349-B2 Glucosylceramide synthase inhibitors GENZYME CORPORATION (US) 2024-08-13 US disclosed
CN-112110811-B Preparation method of bilastine intermediate 北京万全德众医药生物技术有限公司 2024-08-13 CN disclosed
EP-4349408-A2 METHODS FOR TREATING PROTEINOPATHIES Genzyme Corporation (US) 2024-04-10 EP disclosed
EP-3267983-B1 METHODS FOR TREATING PROTEINOPATHIES GENZYME CORP (US) 2023-12-20 EP disclosed
CN-107567443-B Biaryl derivatives as GPR120 agonists 株式会社LG化学 2023-04-28 CN disclosed
CN-115925679-A Biaryl derivatives as GPR120 agonists 株式会社LG化学 2023-04-07 CN disclosed
EP-1856058-A2 PHTHALAZINE, AZA- AND DIAZA-PHTHALAZINE COMPOUNDS AND METHODS OF USE Amgen Inc. (US) 2007-11-21 EP disclosed
US-20070179186-A1 for the treatment of non-insulin dependent type 2 diabetes, insulin resistance, obesity, lipid disorders, metabolic syndrome and conditions because of excessive glucocorticoid action; E-4-(2-methyl-2-phenoxy-propionylamino)-adamantane-1-carboxylic acid amide ABBVIE INC. 2007-08-02 US disclosed
US-7217838-B2 Compounds such as E-4-{[1-(4-Chloro-phenyl)-cyclobutanecarbonyl]-amino}-adamantane-1-carboxylic acid; fortherapy of non-insulin dependent type 2 diabetes, insulin resistance, obesity, lipid disorders, metabolic syndrome and diseases and conditions that are mediated by excessive glucocorticoid action ABBOTT LABORATORIES (US) 2007-05-15 US disclosed
WO-2006094187-A2 PHTHALAZINE, AZA- AND DIAZA-PHTHALAZINE COMPOUNDS AND METHODS OF USE AMGEN INC (US) 2006-09-08 WO disclosed
US-20060199817-A1 Phthalazine, aza- and diaza-phthalazine compounds and methods of use AMGEN INC. (US) 2006-09-07 US disclosed
US-20060149070-A1 Compounds such as E-4-{[1-(4-Chloro-phenyl)-cyclobutanecarbonyl]-amino}-adamantane-1-carboxylic acid, for therapy of non-insulin dependent type 2 diabetes, insulin resistance, obesity, lipid disorders, metabolic syndrome and diseases and conditions that are mediated by excessive glucocorticoid action ABBVIE INC. 2006-07-06 US disclosed
US-6043284-A ACYL COENZYME A: CHOLESTEROL ACYLTRANSFERASE (ACAT) INHIBITORS GLAXO WELLCOME INC. (US) 2000-03-28 US disclosed
US-5776951-A ANTICHOLESTEROL AGENT GLAXO WELLCOME INC. (US) 1998-07-07 US disclosed
EP-0706508-A1 ANTI-ATHEROSCLEROTIC DIARYL COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1996-04-17 EP disclosed
WO-1995001326-A1 ANTI-ATHEROSCLEROTIC DIARYL COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1995-01-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070179186-A1 for the treatment of non-insulin dependent type 2 diabetes, insulin resistance, obesity, lipid disorders, metabolic syndrome and conditions because of excessive glucocorticoid action; E-4-(2-methyl-2-phenoxy-propionylamino)-adamantane-1-carboxylic acid amide HSD17B1, HSD3B1, HSD17B2 ALDH1A1 262/4885LMNA 3475/4885NPSR1 1309/4885
US-12527776-B2 Treatment of ciliopathies using inhibitors of glucosylceramide synthase (GCS) GBA1, GBA2, GALC ALDH1A1 1394/4885LMNA 2738/4885NPSR1 1620/4885
US-20060199817-A1 Phthalazine, aza- and diaza-phthalazine compounds and methods of use DAPK2, CDK2, DAPK1 ALDH1A1 1599/4885LMNA 3537/4885NPSR1 1507/4885
US-20060149070-A1 Compounds such as E-4-{[1-(4-Chloro-phenyl)-cyclobutanecarbonyl]-amino}-adamantane-1-carboxylic acid, for therapy of non-insulin dependent type 2 diabetes, insulin resistance, obesity, lipid disorders, metabolic syndrome and diseases and conditions that are mediated by excessive glucocorticoid action HSD17B1, HSD11B1, HSD3B1 ALDH1A1 229/4885LMNA 3850/4885NPSR1 1603/4885
US-12083115-B2 Methods for treating neurological symptoms associated with lysosomal storage diseases GBA1, GBA2, CLN6 ALDH1A1 3359/4885LMNA 242/4885NPSR1 1341/4885
US-12060349-B2 Glucosylceramide synthase inhibitors GBA1, GBA2, GALC ALDH1A1 2066/4885LMNA 2655/4885NPSR1 1562/4885
US-20250026749-A1 GLUCOSYLCERAMIDE SYNTHASE INHIBITORS GBA1, GBA2, GAA ALDH1A1 2144/4885LMNA 2630/4885NPSR1 1896/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.