SCHEMBL9213895

SCHEMBL9213895

COc1cccnc1N1CCN(CCc2c[nH]c3ccc(Cl)cc23)CC1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.59
HTR6 P50406 3/20 0.59
HTR1A P08908 6/20 0.58
HTR7 P34969 2/20 0.52
SLC6A4 P31645 1/20 0.52
IDO1 P14902 1/20 0.50
DRD2 P14416 1/20 0.49
DRD4 P21917 1/20 0.49
DRD3 P35462 1/20 0.49
HTR2A P28223 2/20 0.49
MPO P05164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9211546 0.90 HTR2A (0.64) HTR1ADRD2DRD4DRD3HTR2A
SCHEMBL9214152 0.90 HTR1A (0.65) KCNH2HTR6HTR1AHTR7SLC6A4
SCHEMBL9205321 0.88 DRD2 (0.52) KCNH2HTR6HTR1AHTR7SLC6A4
SCHEMBL9205349 0.87 ABCC1 (0.57) KCNH2HTR6HTR1AHTR7SLC6A4
SCHEMBL9205705 0.84 HTR1A (0.73) KCNH2HTR6HTR1AHTR7SLC6A4
SCHEMBL9274974 0.84 DRD2 (0.57) HTR1ADRD2DRD4DRD3HTR2A
SCHEMBL9210187 0.82 HTR1A (0.64) KCNH2HTR6HTR1AHTR7SLC6A4
SCHEMBL9210900 0.81 HTR1A (0.65) KCNH2HTR6HTR1AHTR7SLC6A4
SCHEMBL6354737 0.81 HTR1A (0.66) KCNH2HTR6HTR1AHTR7SLC6A4
SCHEMBL27989611 0.81 HTR1A (0.69) KCNH2HTR6HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0345808-B1 1-Indolylalkyl-4-(substituted-pyridinyl)piperazines BRISTOL MYERS SQUIBB CO (US) 1995-01-11 EP claimed
US-4954502-A Antidepressants BRISTOL-MYERS SQUIBB COMPANY (US) 1990-09-04 US claimed