SCHEMBL9212261

SCHEMBL9212261

COc1cc2c(cc1OC)CN(CC1CCN(CCCc3cn(C)c4ccccc34)C1)C2

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.49
ALDH1A1 P00352 3/20 0.44
TSHR P16473 1/20 0.44
HTR4 Q13639 1/20 0.42
SLC6A4 P31645 2/20 0.42
HTR1A P08908 1/20 0.42
DRD2 P14416 1/20 0.42
SLC6A2 P23975 1/20 0.42
HTR2A P28223 1/20 0.42
DRD3 P35462 1/20 0.42
SLC6A3 Q01959 1/20 0.42
HTR7 P34969 1/20 0.42
KDM4E B2RXH2 1/20 0.41
TP53 P04637 1/20 0.41
LMNA P02545 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9212347 0.85 ALDH1A1 (0.50) ABCB1ALDH1A1TSHRSLC6A4HTR1A
Hydrochloric Acid SCHEMBL9207604 0.81 HTR1A (0.52) SLC6A4HTR1ADRD2SLC6A2HTR2A
SCHEMBL9213653 0.79 ALDH1A1 (0.45) ABCB1ALDH1A1TSHRSLC6A4HTR2A
SCHEMBL9211758 0.77 PDE4B (0.48) ABCB1DRD3HTR7
SCHEMBL9213552 0.77 ALDH1A1 (0.38) ALDH1A1TSHRSLC6A4HTR1AHTR2A
SCHEMBL9739656 0.76 ALDH1A1 (0.42) ABCB1ALDH1A1TSHRSLC6A4HTR2A
SCHEMBL9206815 0.72 HTR1A (0.55) SLC6A4HTR1ADRD2HTR2ADRD3
SCHEMBL9217614 0.71 ACHE (0.50) ABCB1HTR7KDM4EMEN1KMT2A
SCHEMBL9216571 0.70 PDE4D (0.49) SLC6A4HTR1ADRD2HTR2ADRD3
Hydrochloric Acid SCHEMBL9740012 0.69 PDE4D (0.48) SLC6A4HTR1ADRD2HTR2ADRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed