SCHEMBL9212612

SCHEMBL9212612

CCCNC(=S)Nc1ccc(/C=C/CC(=O)O)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.56
MAPT P10636 5/20 0.55
ALOX12 P18054 3/20 0.55
GAA P10253 3/20 0.55
CYP1A2 P05177 1/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2C19 P33261 1/20 0.54
ALDH1A1 P00352 5/20 0.52
PAM P19021 1/20 0.46
LMNA P02545 6/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
MAOB P27338 1/20 0.43
MEN1 O00255 3/20 0.43
POLB P06746 1/20 0.43
BLM P54132 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
HTT P42858 3/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9213200 0.89 KDM4C (0.49) KMT2AMAPTALOX12GAAALDH1A1
SCHEMBL9210792 0.83 PAM (0.51) KMT2AMAPTGAACYP1A2CYP2C9
SCHEMBL8828415 0.77 PAM (0.58) KMT2AMAPTGAAALDH1A1PAM
SCHEMBL8828409 0.77 PAM (0.58) KMT2AMAPTGAAALDH1A1PAM
SCHEMBL7151984 0.75 CYP1A2 (0.68) KMT2AMAPTALOX12GAACYP1A2
SCHEMBL9213867 0.75 PAM (0.54) KMT2AMAPTALDH1A1PAMLMNA
SCHEMBL5458013 0.73 KMT2A (1.00) KMT2AMAPTALOX12GAACYP1A2
SCHEMBL25517525 0.72 CYP1A2 (0.72) KMT2AMAPTALOX12GAACYP1A2
SCHEMBL5455860 0.72 CYP1A2 (0.72) KMT2AMAPTALOX12GAACYP1A2
SCHEMBL9230563 0.72 PAM (0.41) KMT2AMAPTALDH1A1PAMMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0399358-B1 Butenoic acid derivatives EISAI CO LTD (JP) 1995-03-08 EP disclosed
EP-0633248-A1 Butenoic acid derivatives Eisai Co., Ltd. (JP) 1995-01-11 EP disclosed
EP-0589491-A1 Butenoic acid derivatives Eisai Co., Ltd. (JP) 1994-03-30 EP disclosed
EP-0399358-A2 Butenoic acid derivatives Eisai Co., Ltd. (JP) 1990-11-28 EP disclosed