SCHEMBL9212896

SCHEMBL9212896

COc1ccc(OCCCN2CCC(COS(=O)(=O)Cc3ccccc3)C2)cc1OC

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.48
SLC6A2 P23975 1/20 0.47
SLC6A4 P31645 1/20 0.47
MAOB P27338 3/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
LTA4H P09960 2/20 0.44
TMEM97 Q5BJF2 1/20 0.44
SIGMAR1 Q99720 1/20 0.44
ACHE P22303 2/20 0.44
BCHE P06276 1/20 0.44
DRD2 P14416 1/20 0.43
DRD4 P21917 1/20 0.43
ADRA1A P35348 1/20 0.43
ADRA1B P35368 1/20 0.43
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9214315 0.85 ABCB1 (0.56) ABCB1SLC6A4TMEM97SIGMAR1
SCHEMBL9205156 0.84 CHRNB2 (0.54) KMT2ALTA4HKDM4EALDH1A1
SCHEMBL9210505 0.83 HRH3 (0.57) MEN1KMT2AACHEKDM4EALDH1A1
SCHEMBL9212384 0.83 ADRA1A (0.52) MEN1KMT2ALTA4HADRA1AADRA1B
SCHEMBL10648297 0.82 ABCB1 (0.45) ABCB1MEN1KMT2ASIGMAR1DRD2
SCHEMBL9208504 0.76 HRH2 (0.49) KMT2ALTA4HTMEM97SIGMAR1KDM4E
SCHEMBL9739469 0.73 ABCB1 (0.55) ABCB1SLC6A4TMEM97SIGMAR1
SCHEMBL9739220 0.72 HRH3 (0.52) SLC6A2SLC6A4KMT2AKDM4EALDH1A1
SCHEMBL9278988 0.71 HRH3 (0.48)
SCHEMBL9739552 0.71 CHRNB2 (0.57) MEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0410953-B1 Piperidine compounds with glycosidase inhibition activity MONSANTO CO (US) 1995-11-08 EP disclosed
US-5175168-A Glycosidase inhibitors MONSANTO COMPANY (US) 1992-12-29 US disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
US-5025021-A 1,2-dideoxy-2-fluoronojirimycin as glycosidase inhibitors MONSANTO COMPANY (US) 1991-06-18 US disclosed
EP-0410953-A2 Piperidine compounds with glycosidase inhibition activity MONSANTO COMPANY (US) 1991-01-30 EP disclosed