SCHEMBL9739220

SCHEMBL9739220

COc1ccc2cc(OCCCN3CCCC(COS(=O)(=O)c4ccccc4)C3)ccc2c1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 10/20 0.52
CHRNB2 P17787 2/20 0.49
CHRNA4 P43681 2/20 0.49
CHRNB4 P30926 1/20 0.49
CHRNA3 P32297 1/20 0.49
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
KMT2A Q03164 1/20 0.49
SLC6A2 P23975 1/20 0.46
SLC6A4 P31645 1/20 0.46
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45
KDM2B Q8NHM5 1/20 0.44
DRD3 P35462 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9740303 0.93 HRH3 (0.60) HRH3CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL9739552 0.92 CHRNB2 (0.57) HRH3CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL9205099 0.89 HRH3 (0.48) HRH3CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL9211609 0.86 KDM4E (0.55) HRH3CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL9208504 0.86 HRH2 (0.49) HRH3CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL9210505 0.81 HRH3 (0.57) HRH3CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL9205156 0.80 CHRNB2 (0.54) HRH3CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL9212384 0.78 ADRA1A (0.52) KDM4EALDH1A1KMT2ADRD3
SCHEMBL9207731 0.76 SIGMAR1 (0.43) HRH3
SCHEMBL9740178 0.76 HRH3 (0.48) HRH3ALDH1A1KMT2APOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed