SCHEMBL9213112

SCHEMBL9213112

c1ccc(CN2CCNCc3cccc(n3)CNCC2)cc1

nearest known ligand 0.88

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 8/20 0.88
SIGMAR1 Q99720 4/20 0.67
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
ALDH1A1 P00352 1/20 0.49
CYP2C9 P11712 1/20 0.49
TSHR P16473 1/20 0.49
CYP2C19 P33261 1/20 0.49
HIF1A Q16665 1/20 0.49
DRD2 P14416 3/20 0.47
DRD4 P21917 3/20 0.47
DRD3 P35462 3/20 0.47
CHRM2 P08172 1/20 0.45
CHRM1 P11229 1/20 0.45
ADRA2C P18825 1/20 0.45
CCR2 P41597 1/20 0.45
CXCL12 P48061 1/20 0.45
BLM P54132 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
HRH3 Q9Y5N1 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL674043 0.85 CXCR4 (0.83) CXCR4SIGMAR1MEN1KMT2ACHRM2
SCHEMBL29490423 0.85 CXCR4 (0.83) CXCR4SIGMAR1MEN1KMT2ACHRM2
SCHEMBL15502455 0.82 CXCR4 (0.78) CXCR4MEN1KMT2AALDH1A1CYP2C19
SCHEMBL83548 0.81 SIGMAR1 (1.00) CXCR4SIGMAR1MEN1KMT2AALDH1A1
SCHEMBL276363 0.81 SIGMAR1 (1.00) CXCR4SIGMAR1MEN1KMT2AALDH1A1
SCHEMBL6138636 0.81 SIGMAR1 (1.00) CXCR4SIGMAR1MEN1KMT2AALDH1A1
Benzene SCHEMBL27761330 0.81 SIGMAR1 (1.00) CXCR4SIGMAR1MEN1KMT2AALDH1A1
SCHEMBL152631 0.81 SIGMAR1 (1.00) CXCR4SIGMAR1MEN1KMT2AALDH1A1
SCHEMBL13250548 0.80 CXCR4 (0.65) CXCR4SIGMAR1MEN1KMT2ACHRM2
SCHEMBL7573306 0.79 SIGMAR1 (0.96) CXCR4SIGMAR1MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5403572-A Macrocyclic polyaza compounds containing 5 or 6 membered rings, process for producing them and pharmaceutical media containing them SCHERING AKTIENGESELLSCHAFT (DE) 1995-04-04 US disclosed
EP-0352218-B1 Macrocyclic polyaza compounds containing rings with 5 or 6 members, methods for their preparation and pharmaceutical compositions containing same SCHERING AG (DE) 1995-02-22 EP disclosed
US-5334371-A Marcocyclic polyaza bicyclo compounds containing 5 or 6 membered rings, and method for MRI SCHERING AKTIENGESELLSCHAFT (DE) 1994-08-02 US disclosed
EP-0352218-A2 Macrocyclic polyaza compounds containing rings with 5 or 6 members, methods for their preparation and pharmaceutical compositions containing same SCHERING AKTIENGESELLSCHAFT (DE) 1990-01-24 EP disclosed