SCHEMBL276363

SCHEMBL276363

c1ccc(CN2CCNCC2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 1.00
MEN1 O00255 2/20 0.68
KMT2A Q03164 2/20 0.68
ALDH1A1 P00352 1/20 0.68
CYP2C9 P11712 1/20 0.68
TSHR P16473 1/20 0.68
CYP2C19 P33261 1/20 0.68
HIF1A Q16665 1/20 0.68
CXCR4 P61073 9/20 0.64
CHRM2 P08172 1/20 0.63
CHRM1 P11229 1/20 0.63
ADRA2C P18825 1/20 0.63
CCR2 P41597 1/20 0.63
CXCL12 P48061 1/20 0.63
BLM P54132 1/20 0.63
TDP1 Q9NUW8 1/20 0.63
HRH3 Q9Y5N1 1/20 0.63
MC4R P32245 1/20 0.59
DRD4 P21917 1/20 0.57
LMNA P02545 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6138636 1.00 SIGMAR1 (1.00) SIGMAR1MEN1KMT2AALDH1A1CYP2C9
SCHEMBL83548 1.00 SIGMAR1 (1.00) SIGMAR1MEN1KMT2AALDH1A1CYP2C9
Benzene SCHEMBL27761330 1.00 SIGMAR1 (1.00) SIGMAR1MEN1KMT2AALDH1A1CYP2C9
SCHEMBL152631 1.00 SIGMAR1 (1.00) SIGMAR1MEN1KMT2AALDH1A1CYP2C9
SCHEMBL7062479 0.98 SIGMAR1 (0.96) SIGMAR1MEN1KMT2AALDH1A1CYP2C9
SCHEMBL7573306 0.98 SIGMAR1 (0.96) SIGMAR1MEN1KMT2AALDH1A1CYP2C9
Hydrochloric Acid SCHEMBL2223234 0.98 SIGMAR1 (0.96) SIGMAR1MEN1KMT2AALDH1A1CYP2C9
SCHEMBL8145866 0.98 SIGMAR1 (0.96) SIGMAR1MEN1KMT2AALDH1A1CYP2C9
SCHEMBL10063607 0.98 SIGMAR1 (0.96) SIGMAR1MEN1KMT2AALDH1A1CYP2C9
Ammonia Solution, Strong SCHEMBL28172574 0.98 SIGMAR1 (0.96) SIGMAR1MEN1KMT2AALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 334 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118125997-A Pterocarpus stilbene paeonol chalcone amide derivative, preparation method and medical application thereof 安徽中医药大学 2024-06-04 CN claimed
CN-117567303-A Chalcone Mannich base compound, pharmaceutical composition, preparation method and application thereof 安徽中医药大学 2024-02-20 CN claimed
CN-116102565-A Isolamine-containing spirochromone compound and preparation method and application thereof 贵州大学 2023-05-12 CN claimed
CN-113717201-B (+/-) -Marinopyrole A derivative and preparation method and application thereof 植恩生物技术股份有限公司 2022-12-16 CN claimed
CN-115260046-A Abietate compound and preparation method and application thereof 贵州大学 2022-11-01 CN claimed
CN-115141208-A Podophyllotoxin compound containing various ester group structures and preparation method and application thereof 贵州大学 2022-10-04 CN claimed
CN-114920722-A 7-hydroxy-3-acetyl coumarin oxime compound, preparation method and medical application thereof 何黎琴 2022-08-19 CN claimed
CN-113717201-A (+/-) -Marinopyrole A derivative and preparation method and application thereof 植恩生物技术股份有限公司 2021-11-30 CN claimed
CN-112707843-A Novel paeonol oxime compound, preparation method and medical application thereof 何黎琴 2021-04-27 CN claimed
CN-112624931-A Pterostilbene amine compounds containing isopropanol aromatic ether structure and preparation method and application thereof 贵州大学 2021-04-09 CN claimed
US-4409219-A BACTERICIDES EGYT GYOGYSZERVEGYESZETI GYAR (HU) 1983-10-11 US claimed
US-4395413-A NICOTINE ANTIALLERGEN, ANESTHETIC, ANALGESIC, HYPOTENSIVE, AND ANTIULCER AGENT EGYT GYOGYSZERVEGYESZETI GYAR (HU) 1983-07-26 US claimed
EP-0023569-B1 DERIVATIVES OF CARBOXYLIC ACIDS, THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM Dr. Karl Thomae GmbH (DE) 1983-06-22 EP claimed
EP-0022371-B1 SUBSTITUTED PIPERAZINES AND PIPERIDINES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM PFIZER INC. (US) 1983-01-19 EP claimed
US-4342762-A USEFUL AS TRANQUILIZERS, ANALGESICS, ANTIEPILEPTIC AGENTS, AND AS A TREATMENT FOR PARKINSON'S DISEASE EGYT GYOGYSZERVEGYESZETI GYAR (HU) 1982-08-03 US claimed
US-4324786-A SEDATIVES, ANALGESICS, ANTIINFLAMMATORY, ANTIPYRETIC EGYT GYOGYSZERVEGYESZETI GYAR (HU) 1982-04-13 US claimed
US-4279905-A GASTROINTESTINAL DISORDERS KALI-CHEMIE PHARMA GMBH (DE) 1981-07-21 US claimed
EP-0025109-A2 1-Benzoxepin-5(2H)-one derivatives and their salts, and processes for their preparation Kali-Chemie Pharma GmbH (DE) 1981-03-18 EP claimed
EP-0022371-A1 Substituted piperazines and piperidines and pharmaceutical compositions containing them PFIZER INC. (US) 1981-01-14 EP claimed
US-4128643-A 4-Quinazolinyl-guanidines HOECHST AKTIENGESELLSCHAFT (DE) 1978-12-05 US claimed