SCHEMBL9213249

SCHEMBL9213249

COc1cc2c(cc1OC)CC(=O)N(CC1CCCN(CCCc3coc4ccccc34)C1)CC2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.44
CHRNA4 P43681 3/20 0.44
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
HCN4 Q9Y3Q4 2/20 0.40
MAPT P10636 1/20 0.40
CYP3A4 P08684 1/20 0.39
ALOX15 P16050 1/20 0.39
CHRM2 P08172 1/20 0.37
HTR1A P08908 1/20 0.37
SLC6A4 P31645 1/20 0.37
DRD3 P35462 1/20 0.37
KCNH2 Q12809 1/20 0.37
MAOB P27338 2/20 0.37
HRH3 Q9Y5N1 2/20 0.37
GAA P10253 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ABCB1 P08183 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9210130 0.95 CHRNB2 (0.42) CHRNB2CHRNA4CHRNB4CHRNA3HCN4
SCHEMBL9214343 0.91 CHRNB2 (0.39) CHRNB2CHRNA4HTR1AMAOBHRH3
SCHEMBL9216575 0.89 CHRNB2 (0.37) CHRNB2CHRNA4HTR1ADRD3MAOB
SCHEMBL9211008 0.86 CHRNB2 (0.37) CHRNB2CHRNA4HTR1ASLC6A4MEN1
SCHEMBL9215387 0.84 LTA4H (0.37) CHRNB2CHRNA4HTR1ASLC6A4DRD3
Hydrochloric Acid SCHEMBL9741187 0.84 PDE4D (0.48) HTR1ASLC6A4DRD3KCNH2
SCHEMBL9214709 0.82 HCN4 (0.41) CHRNB2CHRNA4CHRNB4CHRNA3HCN4
SCHEMBL9215979 0.82 PDE4D (0.48) HTR1ASLC6A4DRD3SMN1; SMN2
SCHEMBL9210593 0.82 HCN4 (0.40) CHRNB2CHRNA4CHRNB4CHRNA3HCN4
Water SCHEMBL9740391 0.82 PDE4D (0.47) HTR1ASLC6A4DRD3SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed