SCHEMBL9215387

SCHEMBL9215387

O=C1Cc2cc3c(cc2CCN1CC1CCCN(CCc2coc4ccccc24)C1)OCO3

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 2/20 0.37
ALDH1A1 P00352 1/20 0.36
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35
HTR1A P08908 5/20 0.35
PDE2A O00408 1/20 0.34
DRD2 P14416 2/20 0.34
HTR2A P28223 2/20 0.34
DRD3 P35462 2/20 0.34
SIGMAR1 Q99720 1/20 0.34
LMNA P02545 2/20 0.33
SLC6A4 P31645 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9216575 0.95 CHRNB2 (0.37) LTA4HALDH1A1CHRNB2CHRNA4HTR1A
SCHEMBL9211008 0.91 CHRNB2 (0.37) LTA4HCHRNB2CHRNA4HTR1APDE2A
SCHEMBL9210130 0.89 CHRNB2 (0.42) CHRNB2CHRNA4HTR1ADRD3SLC6A4
SCHEMBL9214343 0.86 CHRNB2 (0.39) LTA4HCHRNB2CHRNA4HTR1APDE2A
SCHEMBL9206684 0.85 HTR1A (0.41) LTA4HALDH1A1HTR1APDE2ALMNA
SCHEMBL9213249 0.84 CHRNB2 (0.44) CHRNB2CHRNA4HTR1ADRD3SLC6A4
SCHEMBL9217026 0.84 MAPK1 (0.40) LTA4HALDH1A1PDE2ADRD2LMNA
SCHEMBL9215793 0.82 HTR1A (0.39) LTA4HALDH1A1HTR1APDE2ALMNA
SCHEMBL9739483 0.82 LTA4H (0.42) LTA4HALDH1A1LMNAKDM4EMEN1
SCHEMBL9207563 0.81 LTA4H (0.37) LTA4HALDH1A1LMNAKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed