SCHEMBL9216575

SCHEMBL9216575

O=C1Cc2cc3c(cc2CCN1CC1CCCN(CCCc2coc4ccccc24)C1)OCO3

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.37
CHRNA4 P43681 2/20 0.37
LTA4H P09960 1/20 0.36
ALDH1A1 P00352 1/20 0.36
PDE2A O00408 1/20 0.34
MAOB P27338 2/20 0.33
HRH3 Q9Y5N1 2/20 0.33
DRD2 P14416 2/20 0.33
HTR2A P28223 2/20 0.33
DRD3 P35462 2/20 0.33
PRMT5 O14744 1/20 0.33
WDR77 Q9BQA1 1/20 0.33
HTR1A P08908 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
LMNA P02545 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HTR7 P34969 2/20 0.33
GRM5 P41594 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9215387 0.95 LTA4H (0.37) CHRNB2CHRNA4LTA4HALDH1A1PDE2A
SCHEMBL9214343 0.91 CHRNB2 (0.39) CHRNB2CHRNA4LTA4HPDE2AMAOB
SCHEMBL9213249 0.89 CHRNB2 (0.44) CHRNB2CHRNA4MAOBHRH3DRD3
SCHEMBL9211008 0.86 CHRNB2 (0.37) CHRNB2CHRNA4LTA4HPDE2ADRD2
SCHEMBL9210130 0.84 CHRNB2 (0.42) CHRNB2CHRNA4DRD3HTR1AMEN1
SCHEMBL9216989 0.83 HTR1A (0.36) LTA4HALDH1A1PDE2APRMT5WDR77
SCHEMBL9207818 0.83 HTR1A (0.43) ALDH1A1DRD2HTR2ADRD3HTR1A
SCHEMBL9215741 0.82 HTR1A (0.38) CHRNB2CHRNA4LTA4HALDH1A1PDE2A
Water SCHEMBL9739270 0.82 HTR1A (0.43) ALDH1A1DRD2HTR2ADRD3HTR1A
SCHEMBL9208812 0.82 DRD2 (0.38) LTA4HALDH1A1DRD2DRD3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed