SCHEMBL9211008

SCHEMBL9211008

Cc1cc2c(cc1C)CC(=O)N(CC1CCCN(CCc3coc4ccccc34)C1)CC2

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.37
CHRNA4 P43681 2/20 0.37
PDE2A O00408 1/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
HTR1A P08908 5/20 0.35
CXCR4 P61073 1/20 0.35
SIGMAR1 Q99720 1/20 0.34
LTA4H P09960 1/20 0.34
SLC6A4 P31645 2/20 0.34
LMNA P02545 1/20 0.34
DRD2 P14416 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9214343 0.95 CHRNB2 (0.39) CHRNB2CHRNA4PDE2AHTR1ASIGMAR1
SCHEMBL9210130 0.91 CHRNB2 (0.42) CHRNB2CHRNA4KMT2AMEN1HTR1A
SCHEMBL9215387 0.91 LTA4H (0.37) CHRNB2CHRNA4PDE2AKMT2AMEN1
SCHEMBL9213249 0.86 CHRNB2 (0.44) CHRNB2CHRNA4KMT2AMEN1HTR1A
SCHEMBL9216575 0.86 CHRNB2 (0.37) CHRNB2CHRNA4PDE2AKMT2AMEN1
SCHEMBL9211495 0.83 HTR1A (0.42) PDE2AKMT2AMEN1HTR1ACXCR4
SCHEMBL9215152 0.82 MAPK1 (0.44) PDE2ALTA4HLMNADRD2
SCHEMBL9215232 0.81 HTR1A (0.40) PDE2AKMT2AMEN1HTR1ACXCR4
SCHEMBL9207422 0.80 HRH3 (0.40) KMT2AMEN1CXCR4LTA4HLMNA
SCHEMBL9213117 0.80 MAPK1 (0.42) PDE2ALTA4HLMNADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed